NO326155B1 - 2H-pyridazin-3-onderivater, farmasoytiske preparater inneholdende slike og fremgangsmate for fremstilling av den aktive ingrediensen, anvendelse som medikamenter og farmasoytiske preparater - Google Patents

2H-pyridazin-3-onderivater, farmasoytiske preparater inneholdende slike og fremgangsmate for fremstilling av den aktive ingrediensen, anvendelse som medikamenter og farmasoytiske preparater Download PDF

Info

Publication number: NO326155B1
Authority: NO; Norway
Prior art keywords: formula; pyridazin; derivative; acid addition; group
Prior art date: 2001-07-26

Application number

NO20040268A

Other languages

English (en)

Norwegian (no)

Other versions

NO20040268L (no

Inventor

Aniko Miklosne Kovacs

Istvan Gacsalyi

Jozsef Barkoczy

Janos Wellmann

Katalin Pallagi

Peter Kotay Nagy

Gyorgy Levay

Andras Egyed

Gyula Simig

Judit Raczne Bajnogel

Eva Schmidt

Gabor Szenasi

Original Assignee

Egyt Gyogyszervegyeszeti Gyar

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-07-26

Filing date

2004-01-20

Publication date

2008-10-13

2004-01-20 Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar

2004-03-23 Publication of NO20040268L publication Critical patent/NO20040268L/no

2008-10-13 Publication of NO326155B1 publication Critical patent/NO326155B1/no

Links

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239000001506 calcium phosphate Substances 0.000 description 1
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KVWDHTXUZHCGIO-UHFFFAOYSA-N olanzapine Chemical compound C1CN(C)CCN1C1=NC2=CC=CC=C2NC2=C1C=C(C)S2 KVWDHTXUZHCGIO-UHFFFAOYSA-N 0.000 description 1
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ZTHJULTYCAQOIJ-WXXKFALUSA-N quetiapine fumarate Chemical compound [H+].[H+].[O-]C(=O)\C=C\C([O-])=O.C1CN(CCOCCO)CCN1C1=NC2=CC=CC=C2SC2=CC=CC=C12.C1CN(CCOCCO)CCN1C1=NC2=CC=CC=C2SC2=CC=CC=C12 ZTHJULTYCAQOIJ-WXXKFALUSA-N 0.000 description 1
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238000010992 reflux Methods 0.000 description 1
230000001850 reproductive effect Effects 0.000 description 1
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229940035004 seroquel Drugs 0.000 description 1
229910000030 sodium bicarbonate Inorganic materials 0.000 description 1
235000017557 sodium bicarbonate Nutrition 0.000 description 1
229910000029 sodium carbonate Inorganic materials 0.000 description 1
239000011780 sodium chloride Substances 0.000 description 1
235000019333 sodium laurylsulphate Nutrition 0.000 description 1
239000002904 solvent Substances 0.000 description 1
239000001593 sorbitan monooleate Substances 0.000 description 1
235000011069 sorbitan monooleate Nutrition 0.000 description 1
229940035049 sorbitan monooleate Drugs 0.000 description 1
239000000600 sorbitol Substances 0.000 description 1
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239000008107 starch Substances 0.000 description 1
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Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

NO20040268A 2001-07-26 2004-01-20 2H-pyridazin-3-onderivater, farmasoytiske preparater inneholdende slike og fremgangsmate for fremstilling av den aktive ingrediensen, anvendelse som medikamenter og farmasoytiske preparater NO326155B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
HU0103063A HU225955B1 (en)	2001-07-26	2001-07-26	Novel 2h-pyridazin-3-one derivatives, process for their preparation, their use and pharmaceutical compositions containing them
PCT/HU2002/000072 WO2003010166A1 (en)	2001-07-26	2002-07-24	Novel 2h-pyridazine-3-one derivatives, pharmaceutical compositions containing the same and a process for the preparation of the active ingredient

Publications (2)

Publication Number	Publication Date
NO20040268L NO20040268L (no)	2004-03-23
NO326155B1 true NO326155B1 (no)	2008-10-13

Family

ID=89979562

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20040268A NO326155B1 (no)	2001-07-26	2004-01-20	2H-pyridazin-3-onderivater, farmasoytiske preparater inneholdende slike og fremgangsmate for fremstilling av den aktive ingrediensen, anvendelse som medikamenter og farmasoytiske preparater

Country Status (28)

Country	Link
US (1)	US7098210B2 (zh)
EP (1)	EP1417206B1 (zh)
JP (1)	JP4249012B2 (zh)
KR (1)	KR100909514B1 (zh)
CN (1)	CN1247571C (zh)
AR (2)	AR036248A1 (zh)
AT (1)	ATE466859T1 (zh)
AU (1)	AU2002321669B8 (zh)
BR (1)	BR0211440A (zh)
CA (1)	CA2453917C (zh)
CY (1)	CY1110240T1 (zh)
CZ (1)	CZ2004123A3 (zh)
DE (1)	DE60236294D1 (zh)
DK (1)	DK1417206T3 (zh)
EA (1)	EA006246B1 (zh)
ES (1)	ES2345541T3 (zh)
HK (1)	HK1067626A1 (zh)
HU (1)	HU225955B1 (zh)
MA (1)	MA27867A1 (zh)
MX (1)	MXPA04000814A (zh)
NO (1)	NO326155B1 (zh)
NZ (1)	NZ531154A (zh)
PL (1)	PL206824B1 (zh)
PT (1)	PT1417206E (zh)
SI (1)	SI1417206T1 (zh)
SK (1)	SK552004A3 (zh)
WO (1)	WO2003010166A1 (zh)
ZA (1)	ZA200400482B (zh)

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HU227255B1 (en) *	2002-04-26	2010-12-28	Egis Gyogyszergyar Nyilvanosan Muekoedoe Reszvenytarsasag	Novel piperidine-alkyl-amino-pyridazine derivatives, pharmaceutical compositions containing the same and process for the preparation of the active ingredient
US7852298B2 (en)	2005-06-08	2010-12-14	Ignis Innovation Inc.	Method and system for driving a light emitting device display
US9489891B2 (en)	2006-01-09	2016-11-08	Ignis Innovation Inc.	Method and system for driving an active matrix display circuit
EP1971975B1 (en)	2006-01-09	2015-10-21	Ignis Innovation Inc.	Method and system for driving an active matrix display circuit
US9269322B2 (en)	2006-01-09	2016-02-23	Ignis Innovation Inc.	Method and system for driving an active matrix display circuit
HUP0600555A3 (en) *	2006-07-03	2008-10-28	Egis Gyogyszergyar Nyrt	Use of 4-chloro-5-{2-[4-(6-fluoro-1,2-benz[d]izoxazol-3-yl)piperidin-1-yl]ethylamino}2-methyl-3(2h)-piridazinon for the production of pharmaceutical compositions for influencing cognitive functions and causing neuroprotective effect
JP5466694B2 (ja)	2008-04-18	2014-04-09	イグニス・イノベーション・インコーポレイテッド	発光デバイス・ディスプレイのためのシステムおよび駆動方法
CA2637343A1 (en)	2008-07-29	2010-01-29	Ignis Innovation Inc.	Improving the display source driver
US9370075B2 (en)	2008-12-09	2016-06-14	Ignis Innovation Inc.	System and method for fast compensation programming of pixels in a display
US8633873B2 (en)	2009-11-12	2014-01-21	Ignis Innovation Inc.	Stable fast programming scheme for displays
CA2687631A1 (en)	2009-12-06	2011-06-06	Ignis Innovation Inc	Low power driving scheme for display applications
CA2696778A1 (en)	2010-03-17	2011-09-17	Ignis Innovation Inc.	Lifetime, uniformity, parameter extraction methods
US9351368B2 (en)	2013-03-08	2016-05-24	Ignis Innovation Inc.	Pixel circuits for AMOLED displays
US20140368491A1 (en)	2013-03-08	2014-12-18	Ignis Innovation Inc.	Pixel circuits for amoled displays
US9886899B2 (en)	2011-05-17	2018-02-06	Ignis Innovation Inc.	Pixel Circuits for AMOLED displays
JP2014522506A (ja)	2011-05-28	2014-09-04	イグニス・イノベイション・インコーポレーテッド	ディスプレイのピクセルの速い補償プログラミングためのシステムと方法
US9747834B2 (en)	2012-05-11	2017-08-29	Ignis Innovation Inc.	Pixel circuits including feedback capacitors and reset capacitors, and display systems therefore
US9786223B2 (en)	2012-12-11	2017-10-10	Ignis Innovation Inc.	Pixel circuits for AMOLED displays
US9336717B2 (en)	2012-12-11	2016-05-10	Ignis Innovation Inc.	Pixel circuits for AMOLED displays
WO2014124755A1 (de)	2013-02-18	2014-08-21	Jürgen Von Der Ohe	Verfahren und vorrichtung zum kaltstrahlreinigen
CA2894717A1 (en)	2015-06-19	2016-12-19	Ignis Innovation Inc.	Optoelectronic device characterization in array with shared sense line
US9721505B2 (en)	2013-03-08	2017-08-01	Ignis Innovation Inc.	Pixel circuits for AMOLED displays
CA2873476A1 (en)	2014-12-08	2016-06-08	Ignis Innovation Inc.	Smart-pixel display architecture
CA2886862A1 (en)	2015-04-01	2016-10-01	Ignis Innovation Inc.	Adjusting display brightness for avoiding overheating and/or accelerated aging
US10657895B2 (en)	2015-07-24	2020-05-19	Ignis Innovation Inc.	Pixels and reference circuits and timing techniques
US10373554B2 (en)	2015-07-24	2019-08-06	Ignis Innovation Inc.	Pixels and reference circuits and timing techniques
CA2898282A1 (en)	2015-07-24	2017-01-24	Ignis Innovation Inc.	Hybrid calibration of current sources for current biased voltage progra mmed (cbvp) displays
CA2908285A1 (en)	2015-10-14	2017-04-14	Ignis Innovation Inc.	Driver with multiple color pixel structure

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IE62890B1 (en) *	1988-12-06	1995-03-08	Hafslund Nycomed Pharma	New piperazinylalkyl-3(2h)-pyridazinones process for the preparation thereof and the use thereof as agents lowering blood pressure
IL117646A (en) *	1995-04-12	2000-06-01	Ferrer Int	7-¬3-¬4-(6-fluoro-1,2-benzisoxazole-3-YL)piperidin-1-YL¾propoxy¾3-alkyl-chromen-4-ones their preparation their uses and pharmaceutical compositions comprising them

2001
- 2001-07-26 HU HU0103063A patent/HU225955B1/hu not_active IP Right Cessation
2002
- 2002-07-24 JP JP2003515525A patent/JP4249012B2/ja not_active Expired - Fee Related
- 2002-07-24 DE DE60236294T patent/DE60236294D1/de not_active Expired - Lifetime
- 2002-07-24 EA EA200400223A patent/EA006246B1/ru not_active IP Right Cessation
- 2002-07-24 KR KR1020047001151A patent/KR100909514B1/ko active IP Right Grant
- 2002-07-24 PT PT02755381T patent/PT1417206E/pt unknown
- 2002-07-24 SK SK55-2004A patent/SK552004A3/sk unknown
- 2002-07-24 EP EP02755381A patent/EP1417206B1/en not_active Expired - Lifetime
- 2002-07-24 WO PCT/HU2002/000072 patent/WO2003010166A1/en active IP Right Grant
- 2002-07-24 AT AT02755381T patent/ATE466859T1/de active
- 2002-07-24 DK DK02755381.7T patent/DK1417206T3/da active
- 2002-07-24 AU AU2002321669A patent/AU2002321669B8/en not_active Ceased
- 2002-07-24 MX MXPA04000814A patent/MXPA04000814A/es active IP Right Grant
- 2002-07-24 NZ NZ531154A patent/NZ531154A/en not_active IP Right Cessation
- 2002-07-24 US US10/484,619 patent/US7098210B2/en not_active Expired - Fee Related
- 2002-07-24 SI SI200230914T patent/SI1417206T1/sl unknown
- 2002-07-24 BR BR0211440-2A patent/BR0211440A/pt active Search and Examination
- 2002-07-24 CN CNB028163737A patent/CN1247571C/zh not_active Expired - Fee Related
- 2002-07-24 CA CA002453917A patent/CA2453917C/en not_active Expired - Fee Related
- 2002-07-24 PL PL367447A patent/PL206824B1/pl unknown
- 2002-07-24 ES ES02755381T patent/ES2345541T3/es not_active Expired - Lifetime
- 2002-07-24 CZ CZ2004123A patent/CZ2004123A3/cs unknown
- 2002-07-26 AR ARP020102834A patent/AR036248A1/es not_active Application Discontinuation
2004
- 2004-01-19 MA MA27487A patent/MA27867A1/fr unknown
- 2004-01-20 NO NO20040268A patent/NO326155B1/no not_active IP Right Cessation
- 2004-01-22 ZA ZA2004/00482A patent/ZA200400482B/en unknown
- 2004-11-12 HK HK04108974.9A patent/HK1067626A1/xx unknown
2010
- 2010-07-22 CY CY20101100690T patent/CY1110240T1/el unknown
2012
- 2012-11-08 AR ARP120104216A patent/AR088808A2/es unknown

Also Published As

Publication number	Publication date
DE60236294D1 (de)	2010-06-17
AR088808A2 (es)	2014-07-10
CA2453917C (en)	2009-06-23
ATE466859T1 (de)	2010-05-15
DK1417206T3 (da)	2010-08-16
EP1417206B1 (en)	2010-05-05
AR036248A1 (es)	2004-08-25
HU225955B1 (en)	2008-01-28
EP1417206A1 (en)	2004-05-12
PT1417206E (pt)	2010-07-29
MXPA04000814A (es)	2004-05-21
WO2003010166A1 (en)	2003-02-06
EA006246B1 (ru)	2005-10-27
CY1110240T1 (el)	2015-01-14
ES2345541T3 (es)	2010-09-27
KR100909514B1 (ko)	2009-07-27
HK1067626A1 (en)	2005-04-15
NZ531154A (en)	2005-09-30
KR20040030862A (ko)	2004-04-09
AU2002321669B2 (en)	2008-05-15
CN1545513A (zh)	2004-11-10
PL206824B1 (pl)	2010-09-30
JP4249012B2 (ja)	2009-04-02
NO20040268L (no)	2004-03-23
US7098210B2 (en)	2006-08-29
AU2002321669A2 (en)	2003-02-17
BR0211440A (pt)	2004-07-20
EA200400223A1 (ru)	2004-12-30
AU2002321669B8 (en)	2008-06-05
HUP0103063A2 (hu)	2003-02-28
HUP0103063A3 (en)	2005-06-28
SI1417206T1 (sl)	2010-09-30
MA27867A1 (fr)	2006-05-02
HU0103063D0 (en)	2001-10-28
ZA200400482B (en)	2005-05-25
US20040171619A1 (en)	2004-09-02
PL367447A1 (en)	2005-02-21
CZ2004123A3 (cs)	2004-05-12
CN1247571C (zh)	2006-03-29
CA2453917A1 (en)	2003-02-06
JP2004538293A (ja)	2004-12-24
SK552004A3 (en)	2004-08-03

Legal Events

Date	Code	Title	Description
2018-02-26	MM1K	Lapsed by not paying the annual fees

Publication	Publication Date	Title
NO326155B1 (no)	2008-10-13	2H-pyridazin-3-onderivater, farmasoytiske preparater inneholdende slike og fremgangsmate for fremstilling av den aktive ingrediensen, anvendelse som medikamenter og farmasoytiske preparater
AU2002321669A1 (en)	2003-05-29	Novel 2H-pyridazine-3-one derivatives, pharmaceutical compositions containing the same and a process for the preparation of the active ingredient
JP4485353B2 (ja)	2010-06-23	有効な抗ヒスタミン剤および抗アレルギー剤としての新規インドリルピペリジン誘導体
EA015813B1 (ru)	2011-12-30	Замещенные производные оксадиазола в качестве положительных аллостерических модуляторов метаботропных глутаматных рецепторов
BG61120B2 (bg)	1996-11-29	Производни на 1,2,5,6-тетрахидропиридин-3-карбоксалдехид оксим,метод за получаването им,приложението им като лекарствени средства и съдържащите ги състави
PT811622E (pt)	2000-08-31	Derivados do 3-(piperid-4-il)-1,2-benzisoxazol e do 3-(piperazin-4-il)-1,2-benzisoxazol processos para a sua preparacao e composicoes farmaceuticas que os contem
JP2003501424A (ja)	2003-01-14	抗ヒスタミンおよび抗アレルギー剤としてのインドリルピペリジン誘導体
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