NO321576B1 - Nye morfolinderivater, fremgangsmater for fremstilling derav, anvendelser derav, og farmasoytiske preparater og medikamenter inneholdende de nevnte derivater. - Google Patents

Nye morfolinderivater, fremgangsmater for fremstilling derav, anvendelser derav, og farmasoytiske preparater og medikamenter inneholdende de nevnte derivater. Download PDF

Info

Publication number: NO321576B1
Authority: NO; Norway
Prior art keywords: compound; formula; mixture; methyl; salts
Prior art date: 1999-03-25

Application number

NO20014632A

Other languages

English (en)

Norwegian (no)

Other versions

NO20014632L (no

NO20014632D0 (no

Inventor

Patrick Gueule

Vincenzo Proietto

Xavier Emonds-Alt

Jean Philippe Ducoux

Original Assignee

Sanofi Aventis

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-03-25

Filing date

2001-09-24

Publication date

2006-06-06

2001-09-24 Application filed by Sanofi Aventis filed Critical Sanofi Aventis

2001-09-24 Publication of NO20014632D0 publication Critical patent/NO20014632D0/no

2001-11-26 Publication of NO20014632L publication Critical patent/NO20014632L/no

2006-06-06 Publication of NO321576B1 publication Critical patent/NO321576B1/no

Links

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235000019333 sodium laurylsulphate Nutrition 0.000 description 1
239000004296 sodium metabisulphite Substances 0.000 description 1
235000010262 sodium metabisulphite Nutrition 0.000 description 1
229910052938 sodium sulfate Inorganic materials 0.000 description 1
235000011152 sodium sulphate Nutrition 0.000 description 1
230000000392 somatic effect Effects 0.000 description 1
235000019337 sorbitan trioleate Nutrition 0.000 description 1
229960000391 sorbitan trioleate Drugs 0.000 description 1
241000894007 species Species 0.000 description 1
238000001228 spectrum Methods 0.000 description 1
208000020431 spinal cord injury Diseases 0.000 description 1
208000005198 spinal stenosis Diseases 0.000 description 1
239000008107 starch Substances 0.000 description 1
235000019698 starch Nutrition 0.000 description 1
229940032147 starch Drugs 0.000 description 1
239000008117 stearic acid Substances 0.000 description 1
230000000638 stimulation Effects 0.000 description 1
201000009032 substance abuse Diseases 0.000 description 1
231100000736 substance abuse Toxicity 0.000 description 1
208000011117 substance-related disease Diseases 0.000 description 1
239000005720 sucrose Substances 0.000 description 1
HIFJUMGIHIZEPX-UHFFFAOYSA-N sulfuric acid;sulfur trioxide Chemical compound O=S(=O)=O.OS(O)(=O)=O HIFJUMGIHIZEPX-UHFFFAOYSA-N 0.000 description 1
YBBRCQOCSYXUOC-UHFFFAOYSA-N sulfuryl dichloride Chemical compound ClS(Cl)(=O)=O YBBRCQOCSYXUOC-UHFFFAOYSA-N 0.000 description 1
239000000829 suppository Substances 0.000 description 1
230000001629 suppression Effects 0.000 description 1
239000000375 suspending agent Substances 0.000 description 1
239000012730 sustained-release form Substances 0.000 description 1
208000024891 symptom Diseases 0.000 description 1
239000000454 talc Substances 0.000 description 1
229910052623 talc Inorganic materials 0.000 description 1
125000005931 tert-butyloxycarbonyl group Chemical group [H]C([H])([H])C(OC(*)=O)(C([H])([H])[H])C([H])([H])[H] 0.000 description 1
150000003512 tertiary amines Chemical class 0.000 description 1
230000001225 therapeutic effect Effects 0.000 description 1
238000002560 therapeutic procedure Methods 0.000 description 1
238000011200 topical administration Methods 0.000 description 1
231100000419 toxicity Toxicity 0.000 description 1
230000001988 toxicity Effects 0.000 description 1
239000003053 toxin Substances 0.000 description 1
231100000765 toxin Toxicity 0.000 description 1
108700012359 toxins Proteins 0.000 description 1
ODLHGICHYURWBS-LKONHMLTSA-N trappsol cyclo Chemical compound CC(O)COC[C@H]([C@H]([C@@H]([C@H]1O)O)O[C@H]2O[C@@H]([C@@H](O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O3)[C@H](O)[C@H]2O)COCC(O)C)O[C@@H]1O[C@H]1[C@H](O)[C@@H](O)[C@@H]3O[C@@H]1COCC(C)O ODLHGICHYURWBS-LKONHMLTSA-N 0.000 description 1
230000000472 traumatic effect Effects 0.000 description 1
CYRMSUTZVYGINF-UHFFFAOYSA-N trichlorofluoromethane Chemical compound FC(Cl)(Cl)Cl CYRMSUTZVYGINF-UHFFFAOYSA-N 0.000 description 1
229940029284 trichlorofluoromethane Drugs 0.000 description 1
UFTFJSFQGQCHQW-UHFFFAOYSA-N triformin Chemical compound O=COCC(OC=O)COC=O UFTFJSFQGQCHQW-UHFFFAOYSA-N 0.000 description 1
206010044652 trigeminal neuralgia Diseases 0.000 description 1
229910052722 tritium Inorganic materials 0.000 description 1
231100000397 ulcer Toxicity 0.000 description 1
208000026533 urinary bladder disease Diseases 0.000 description 1
230000024883 vasodilation Effects 0.000 description 1
231100000889 vertigo Toxicity 0.000 description 1
208000027491 vestibular disease Diseases 0.000 description 1
230000003612 virological effect Effects 0.000 description 1
230000009278 visceral effect Effects 0.000 description 1
208000009935 visceral pain Diseases 0.000 description 1
238000005550 wet granulation Methods 0.000 description 1
239000000080 wetting agent Substances 0.000 description 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A61P25/10—Antiepileptics; Anticonvulsants for petit-mal
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Pain & Pain Management (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Pulmonology (AREA)
Urology & Nephrology (AREA)
Rheumatology (AREA)
Otolaryngology (AREA)
Psychiatry (AREA)
Immunology (AREA)
Hospice & Palliative Care (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Dermatology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Plural Heterocyclic Compounds (AREA)

NO20014632A 1999-03-25 2001-09-24 Nye morfolinderivater, fremgangsmater for fremstilling derav, anvendelser derav, og farmasoytiske preparater og medikamenter inneholdende de nevnte derivater. NO321576B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9903854A FR2791346B3 (fr)	1999-03-25	1999-03-25	Nouveaux derives de morpholine, procede pour leur preparation et compositions pharmaceutiques les contenant
PCT/FR2000/000695 WO2000058292A1 (fr)	1999-03-25	2000-03-21	Nouveaux derives de morpholine, procede pour leur preparation et compositions pharmaceutiques les contenant

Publications (3)

Publication Number	Publication Date
NO20014632D0 NO20014632D0 (no)	2001-09-24
NO20014632L NO20014632L (no)	2001-11-26
NO321576B1 true NO321576B1 (no)	2006-06-06

Family

ID=9543720

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20014632A NO321576B1 (no)	1999-03-25	2001-09-24	Nye morfolinderivater, fremgangsmater for fremstilling derav, anvendelser derav, og farmasoytiske preparater og medikamenter inneholdende de nevnte derivater.

Country Status (41)

Country	Link
US (1)	US6506750B1 (de)
EP (1)	EP1165528B1 (de)
JP (1)	JP3853155B2 (de)
KR (1)	KR100696340B1 (de)
CN (1)	CN100422160C (de)
AR (1)	AR023139A1 (de)
AT (1)	ATE275136T1 (de)
AU (1)	AU756855B2 (de)
BG (1)	BG64623B1 (de)
BR (1)	BR0009281B1 (de)
CA (1)	CA2366829C (de)
CO (1)	CO5160340A1 (de)
CZ (1)	CZ300911B6 (de)
DE (1)	DE60013418T2 (de)
DK (1)	DK1165528T3 (de)
EE (1)	EE04525B1 (de)
ES (1)	ES2226794T3 (de)
FR (1)	FR2791346B3 (de)
HK (1)	HK1042092B (de)
HR (1)	HRP20010704B1 (de)
HU (1)	HUP0201863A3 (de)
ID (1)	ID29871A (de)
IL (2)	IL145041A0 (de)
IS (1)	IS2338B (de)
ME (2)	ME00057B (de)
MX (1)	MXPA01009643A (de)
NO (1)	NO321576B1 (de)
NZ (1)	NZ513674A (de)
PE (1)	PE20001596A1 (de)
PL (1)	PL205318B1 (de)
PT (1)	PT1165528E (de)
RS (1)	RS50085B (de)
RU (1)	RU2222537C2 (de)
SI (1)	SI1165528T1 (de)
SK (1)	SK286977B6 (de)
TR (1)	TR200102639T2 (de)
TW (1)	TW534906B (de)
UA (1)	UA73931C2 (de)
UY (1)	UY26079A1 (de)
WO (1)	WO2000058292A1 (de)
ZA (1)	ZA200106981B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2234929T3 (es) *	2000-11-28	2005-07-01	Smithkline Beecham Plc	Derivados de morfolina como antagonistas de los receptores de orexina.
FR2824828B1 (fr) *	2001-05-21	2005-05-20	Sanofi Synthelabo	Nouveaux derives de piperidinecarboxamide, un procede pour leur preparation et les compositions pharmaceutiques les contenant
GB0228787D0 (en) *	2002-12-10	2003-01-15	Pfizer Ltd	Morpholine dopamine agonists
JP2006511555A (ja) *	2002-12-13	2006-04-06	スミスクラインビーチャムコーポレーション	Ｃｃｒ５拮抗剤としての複素環式化合物
JO2485B1 (en) *	2002-12-23	2009-01-20	شركة جانسين فارماسوتيكا ان. في	1-Piperidine-3-Yl-4-Piperidine-4-Yl-Piperazine derivatives substituted and used as quinine antagonists
AR046769A1 (es) *	2003-12-22	2005-12-21	Schering Corp	Composiciones farmaceuticas
FR2873373B1 (fr) *	2004-07-23	2006-09-08	Sanofi Synthelabo	Derives de 4-arylmorpholin-3-one, leur preparation et leur application en therapeutique
CN103142569B (zh) *	2013-02-27	2016-01-20	南京医科大学	2,6-二异丙基苯甲酸及其衍生物作为神经保护剂的应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CZ3134U1 (cs) *	1995-01-10	1995-03-17	Pavel Ing. Janda	Rotor universálního radiálního ventilátoru
FR2729954B1 (fr)	1995-01-30	1997-08-01	Sanofi Sa	Composes heterocycliques substitues, procede pour leur preparation et compositions pharmaceutiques les contenant
US5780466A (en) *	1995-01-30	1998-07-14	Sanofi	Substituted heterocyclic compounds method of preparing them and pharmaceutical compositions in which they are present
RU2135494C1 (ru) *	1995-12-01	1999-08-27	Санкио Компани Лимитед	Гетероциклические соединения и композиция на их основе, проявляющая антагонистическое действие в отношении рецепторов тахикинина
JP3192631B2 (ja) *	1997-05-28	2001-07-30	三共株式会社	飽和複素環化合物からなる医薬
CA2312770A1 (en) *	1997-12-04	1999-06-10	Takahide Nishi	Alicyclic acylated heterocyclic derivatives

1999
- 1999-03-25 FR FR9903854A patent/FR2791346B3/fr not_active Expired - Lifetime
2000
- 2000-03-21 PT PT00911009T patent/PT1165528E/pt unknown
- 2000-03-21 KR KR1020017012121A patent/KR100696340B1/ko not_active IP Right Cessation
- 2000-03-21 BR BRPI0009281-9A patent/BR0009281B1/pt not_active IP Right Cessation
- 2000-03-21 RS YUP-682/01A patent/RS50085B/sr unknown
- 2000-03-21 SI SI200030536T patent/SI1165528T1/xx unknown
- 2000-03-21 CZ CZ20013365A patent/CZ300911B6/cs not_active IP Right Cessation
- 2000-03-21 ME MEP-2008-120A patent/ME00057B/me unknown
- 2000-03-21 EP EP00911009A patent/EP1165528B1/de not_active Expired - Lifetime
- 2000-03-21 SK SK1346-2001A patent/SK286977B6/sk not_active IP Right Cessation
- 2000-03-21 IL IL14504100A patent/IL145041A0/xx unknown
- 2000-03-21 PL PL351317A patent/PL205318B1/pl not_active IP Right Cessation
- 2000-03-21 DK DK00911009T patent/DK1165528T3/da active
- 2000-03-21 CN CNB008055084A patent/CN100422160C/zh not_active Expired - Fee Related
- 2000-03-21 AT AT00911009T patent/ATE275136T1/de active
- 2000-03-21 US US09/937,279 patent/US6506750B1/en not_active Expired - Lifetime
- 2000-03-21 DE DE60013418T patent/DE60013418T2/de not_active Expired - Lifetime
- 2000-03-21 HU HU0201863A patent/HUP0201863A3/hu unknown
- 2000-03-21 NZ NZ513674A patent/NZ513674A/en not_active IP Right Cessation
- 2000-03-21 ES ES00911009T patent/ES2226794T3/es not_active Expired - Lifetime
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- 2000-03-21 WO PCT/FR2000/000695 patent/WO2000058292A1/fr active IP Right Grant
- 2000-03-21 MX MXPA01009643A patent/MXPA01009643A/es unknown
- 2000-03-21 AU AU33016/00A patent/AU756855B2/en not_active Ceased
- 2000-03-21 TR TR2001/02639T patent/TR200102639T2/xx unknown
- 2000-03-21 EE EEP200100499A patent/EE04525B1/xx not_active IP Right Cessation
- 2000-03-21 ID IDW00200101969A patent/ID29871A/id unknown
- 2000-03-21 ME MEP-120/08A patent/MEP12008A/xx unknown
- 2000-03-21 RU RU2001124835/04A patent/RU2222537C2/ru not_active IP Right Cessation
- 2000-03-21 UA UA2001096121A patent/UA73931C2/uk unknown
- 2000-03-21 CA CA002366829A patent/CA2366829C/fr not_active Expired - Lifetime
- 2000-03-23 AR ARP000101299A patent/AR023139A1/es active IP Right Grant
- 2000-03-24 TW TW089105498A patent/TW534906B/zh not_active IP Right Cessation
- 2000-03-24 CO CO00021353A patent/CO5160340A1/es unknown
- 2000-03-27 PE PE2000000258A patent/PE20001596A1/es not_active Application Discontinuation
- 2000-03-27 UY UY26079A patent/UY26079A1/es not_active IP Right Cessation
2001
- 2001-08-21 IL IL145041A patent/IL145041A/en not_active IP Right Cessation
- 2001-08-23 ZA ZA200106981A patent/ZA200106981B/en unknown
- 2001-08-24 IS IS6063A patent/IS2338B/is unknown
- 2001-09-19 BG BG105923A patent/BG64623B1/bg unknown
- 2001-09-24 NO NO20014632A patent/NO321576B1/no not_active IP Right Cessation
- 2001-09-25 HR HR20010704A patent/HRP20010704B1/xx not_active IP Right Cessation
2002
- 2002-05-27 HK HK02103933.2A patent/HK1042092B/zh not_active IP Right Cessation

Also Published As

Publication number	Publication date
AU3301600A (en)	2000-10-16
SK286977B6 (sk)	2009-08-06
PL205318B1 (pl)	2010-04-30
AR023139A1 (es)	2002-09-04
CN100422160C (zh)	2008-10-01
FR2791346B3 (fr)	2001-04-27
WO2000058292A1 (fr)	2000-10-05
ATE275136T1 (de)	2004-09-15
YU68201A (sh)	2004-03-12
HK1042092B (zh)	2005-04-22
KR20010108381A (ko)	2001-12-07
ID29871A (id)	2001-10-18
TW534906B (en)	2003-06-01
CA2366829C (fr)	2007-05-15
JP3853155B2 (ja)	2006-12-06
EP1165528A1 (de)	2002-01-02
ZA200106981B (en)	2002-10-24
TR200102639T2 (tr)	2002-02-21
DK1165528T3 (da)	2005-01-10
FR2791346A1 (fr)	2000-09-29
RS50085B (sr)	2009-01-22
IS6063A (is)	2001-08-24
SI1165528T1 (en)	2005-02-28
AU756855B2 (en)	2003-01-23
NZ513674A (en)	2003-05-30
KR100696340B1 (ko)	2007-03-20
HUP0201863A3 (en)	2003-03-28
JP2002540195A (ja)	2002-11-26
HK1042092A1 (en)	2002-08-02
HRP20010704B1 (en)	2005-04-30
IL145041A0 (en)	2002-06-30
PE20001596A1 (es)	2001-04-01
CZ20013365A3 (cs)	2002-01-16
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Legal Events

Date	Code	Title	Description
2013-10-28	MM1K	Lapsed by not paying the annual fees

Publication	Publication Date	Title
NO321576B1 (no)	2006-06-06	Nye morfolinderivater, fremgangsmater for fremstilling derav, anvendelser derav, og farmasoytiske preparater og medikamenter inneholdende de nevnte derivater.
US6642233B1 (en)	2003-11-04	1-Phenacyl-3-phenyl-3-(piperidylethyl)piperidine derivatives, process for the preparation thereof and pharmaceutical compositions containing them
MXPA03010133A (es)	2005-03-31	Nuevos derivados de piperidinacarboxamida, un procedimiento para su preparacion y las composiciones farmaceuticas que los contienen.
MXPA01008119A (en)	2002-06-05	(1-phenacy-3-phenyl-3-piperidylethyl)piperidine derivatives, method for the production thereof and pharmaceutical compositions containing the same
KR100611262B1 (ko)	2006-08-10	(1-페나시-3-페닐-3-피페리딜에틸)피페리딘 유도체, 그의제조 방법 및 이를 함유하는 제약 조성물
FR2789389A1 (fr)	2000-08-11	Nouveaux derives de piperidine, procede pour leur obtention et compositions pharmaceutiques les contenant
FR2717477A1 (fr)	1995-09-22	Composés antagonistes sélectifs du récepteur NK3 humain et leur utilisation comme médicaments et outils de diagnostic.