NO145951C - Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazolinderivater - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazolinderivater

Info

Publication number: NO145951C
Authority: NO; Norway
Prior art keywords: preparation; therapeutic active; imidazoline derivatives; analogy procedure; active imidazoline
Prior art date: 1976-07-03

Application number

NO772329A

Other languages

English (en)

Other versions

NO772329L (no

NO145951B (no

Inventor

Helmut Staehle

Herbert Koeppe

Werner Kummer

Wolfgang Hoefke

Original Assignee

Boehringer Sohn Ingelheim

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-07-03

Filing date

1977-07-01

Publication date

1982-06-30

1977-07-01 Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim

1978-01-03 Publication of NO772329L publication Critical patent/NO772329L/no

1982-03-22 Publication of NO145951B publication Critical patent/NO145951B/no

1982-06-30 Publication of NO145951C publication Critical patent/NO145951C/no

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Cardiology (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Heart & Thoracic Surgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Electric Clocks (AREA)

NO772329A 1976-07-03 1977-07-01 Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazolinderivater NO145951C (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE2630060A DE2630060C2 (de)	1976-07-03	1976-07-03	2-(2-Brom-6-fluor-phenylimino)-imidazolidin, dessen Säureadditionssalze, diese enthaltende Arzneimittel und Verfahren zu deren Herstellung

Publications (3)

Publication Number	Publication Date
NO772329L NO772329L (no)	1978-01-03
NO145951B NO145951B (no)	1982-03-22
NO145951C true NO145951C (no)	1982-06-30

Family

ID=5982175

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
NO772329A NO145951C (no)	1976-07-03	1977-07-01	Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazolinderivater
NO1994024C NO1994024I1 (no)	1976-07-03	1994-11-25	Romifidin/ 2-brom-6-fluor-N-2-imidazolidinyliden-benzamin og syreaddisjonssalter derav

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
NO1994024C NO1994024I1 (no)	1976-07-03	1994-11-25	Romifidin/ 2-brom-6-fluor-N-2-imidazolidinyliden-benzamin og syreaddisjonssalter derav

Country Status (32)

Country	Link
US (1)	US4166859A (no)
JP (1)	JPS6026108B2 (no)
AT (1)	AT354436B (no)
AU (1)	AU507260B2 (no)
BE (1)	BE856395A (no)
BG (1)	BG28049A3 (no)
CA (1)	CA1088550A (no)
CH (2)	CH633273A5 (no)
CS (1)	CS204005B2 (no)
DD (1)	DD132965A5 (no)
DE (1)	DE2630060C2 (no)
DK (1)	DK146281C (no)
ES (4)	ES460351A1 (no)
FI (1)	FI64146C (no)
FR (1)	FR2356642B1 (no)
GB (1)	GB1575147A (no)
GR (1)	GR63636B (no)
HU (1)	HU180429B (no)
IE (1)	IE45109B1 (no)
IL (1)	IL52433A (no)
LU (1)	LU77679A1 (no)
MX (1)	MX4841E (no)
NL (2)	NL188643C (no)
NO (2)	NO145951C (no)
NZ (1)	NZ184539A (no)
PH (1)	PH14572A (no)
PL (1)	PL102918B1 (no)
PT (1)	PT66756B (no)
SE (1)	SE431871B (no)
SU (2)	SU680644A3 (no)
YU (1)	YU161977A (no)
ZA (1)	ZA773979B (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2806775A1 (de) *	1978-02-17	1979-08-30	Boehringer Sohn Ingelheim	Neue substituierte 2-phenylimino- imidazolidine deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zur herstellung derselben
DE2806811A1 (de) *	1978-02-17	1979-08-23	Boehringer Sohn Ingelheim	Neue substituierte 2-phenylimino- imidazolidine, deren saeureadditionssalze, diese enthaltene arzneimittel und verfahren zur herstellung derselben
US4644007A (en) *	1981-11-20	1987-02-17	Alcon Laboratories, Inc.	3-chloro-4-(4,5-dihydro-1H-imidazo-2-yl)-amino-5-alkylbenzoic acids, esters, salts, compositions and methods
US4517199A (en) *	1981-11-20	1985-05-14	Alcon Laboratories, Inc.	Method for lowering intraocular pressure using phenylimino-imidazoles
US4515800A (en) *	1981-11-20	1985-05-07	Icilio Cavero	Method of lowering intraocular pressure using phenylimino-imidazoles
US4461904A (en) *	1981-11-20	1984-07-24	Alcon Laboratories, Inc.	2-(Trisubstituted phenylimino)-imidazolines
DE3437694A1 (de) *	1984-10-15	1986-04-17	Boehringer Ingelheim Vetmedica GmbH, 6507 Ingelheim	Verwendung einer substanz als sedativum
US4587257A (en) *	1984-12-14	1986-05-06	Alcon Laboratories, Inc.	Control of ocular bleeding using clonidine derivatives
JPH0317363Y2 (no) *	1986-11-19	1991-04-12
US5441339A (en) *	1992-10-22	1995-08-15	Prince Corporation	Vehicle light
WO2005000818A1 (en)	2003-06-27	2005-01-06	Warner-Lambert Company Llc	5-substituted-4-`(substituted phenyl)!amino!-2-pyridone deviatives for use as mek inhibitors
CN115784896A (zh) *	2022-11-24	2023-03-14	山东诚创蓝海医药科技有限公司	一种2-溴-6-氟苯胺的制备方法
CN116063184A (zh) *	2022-12-28	2023-05-05	浙江车头制药股份有限公司	一种2-溴-6-氟苯胺的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1770874B2 (de) *	1968-07-12	1977-09-15	Veb Arzneimittelwerk Dresden, Ddr 8122 Radebeul	Verfahren zur herstellung von 2-(2,6- dichlorphenylamino)-imidazolin-2
BE787683A (fr) *	1971-08-20	1973-02-19	Boehringer Sohn Ingelheim	2-phenylimino-imidazolidines, leurs sels d'addition avec des acides et procedes pour les fabriquer
DE2446758C3 (de) *	1974-10-01	1979-01-04	C.H. Boehringer Sohn, 6507 Ingelheim	2-(2-Fluor-6-trifluormethylphenylimino)-imidazolidin, dessen Säureadditionssalze, Verfahren zur Herstellung dieser Verbindungen und deren Verwendung bei der Bekämpfung der Hypertonie
DE2542702C2 (de) *	1975-09-25	1983-11-10	Lentia GmbH Chem. u. pharm. Erzeugnisse - Industriebedarf, 8000 München	Verfahren zur Herstellung von 1-Benzoyl-2-(2,6-dichlorphenylamino)-2-imidazolin

1976
- 1976-07-03 DE DE2630060A patent/DE2630060C2/de not_active Expired
1977
- 1977-06-20 US US05/808,409 patent/US4166859A/en not_active Expired - Lifetime
- 1977-06-22 AT AT438777A patent/AT354436B/de not_active IP Right Cessation
- 1977-06-23 FI FI771972A patent/FI64146C/fi not_active IP Right Cessation
- 1977-06-30 CH CH807577A patent/CH633273A5/fr not_active IP Right Cessation
- 1977-06-30 YU YU01619/77A patent/YU161977A/xx unknown
- 1977-06-30 AU AU26620/77A patent/AU507260B2/en not_active Expired
- 1977-06-30 CA CA281,884A patent/CA1088550A/en not_active Expired
- 1977-07-01 PH PH19947A patent/PH14572A/en unknown
- 1977-07-01 CS CS774397A patent/CS204005B2/cs unknown
- 1977-07-01 BE BE179022A patent/BE856395A/xx not_active IP Right Cessation
- 1977-07-01 LU LU77679A patent/LU77679A1/xx unknown
- 1977-07-01 MX MX775863U patent/MX4841E/es unknown
- 1977-07-01 GB GB27655/77A patent/GB1575147A/en not_active Expired
- 1977-07-01 GR GR53854A patent/GR63636B/el unknown
- 1977-07-01 PT PT66756A patent/PT66756B/pt unknown
- 1977-07-01 DK DK296477A patent/DK146281C/da active
- 1977-07-01 ZA ZA00773979A patent/ZA773979B/xx unknown
- 1977-07-01 IE IE1371/77A patent/IE45109B1/en not_active IP Right Cessation
- 1977-07-01 FR FR7720343A patent/FR2356642B1/fr not_active Expired
- 1977-07-01 HU HU77BO1672A patent/HU180429B/hu unknown
- 1977-07-01 IL IL52433A patent/IL52433A/xx unknown
- 1977-07-01 NO NO772329A patent/NO145951C/no unknown
- 1977-07-01 JP JP52077979A patent/JPS6026108B2/ja not_active Expired
- 1977-07-01 BG BG036775A patent/BG28049A3/xx unknown
- 1977-07-01 SE SE7707689A patent/SE431871B/xx not_active IP Right Cessation
- 1977-07-01 NL NLAANVRAGE7707308,A patent/NL188643C/xx not_active IP Right Cessation
- 1977-07-01 DD DD7700199844A patent/DD132965A5/xx unknown
- 1977-07-01 SU SU772498148A patent/SU680644A3/ru active
- 1977-07-01 PL PL1977199298A patent/PL102918B1/pl unknown
- 1977-07-01 NZ NZ184539A patent/NZ184539A/xx unknown
- 1977-07-02 ES ES460351A patent/ES460351A1/es not_active Expired
1978
- 1978-02-10 ES ES466850A patent/ES466850A1/es not_active Expired
- 1978-02-10 ES ES466851A patent/ES466851A1/es not_active Expired
- 1978-02-10 ES ES466852A patent/ES466852A1/es not_active Expired
- 1978-03-07 SU SU782589253A patent/SU665800A3/ru active
1981
- 1981-09-02 CH CH566381A patent/CH633275A5/de not_active IP Right Cessation
1993
- 1993-06-29 NL NL930111C patent/NL930111I2/nl unknown
1994
- 1994-11-25 NO NO1994024C patent/NO1994024I1/no unknown

Also Published As

Publication number	Publication date
NL188643C (nl)	1992-08-17
PT66756B (de)	1979-06-07
ATA438777A (de)	1979-06-15
NO772329L (no)	1978-01-03
ES460351A1 (es)	1978-08-16
FR2356642A1 (fr)	1978-01-27
US4166859A (en)	1979-09-04
FI64146C (fi)	1983-10-10
NO1994024I1 (no)	1994-11-25
DD132965A5 (de)	1978-11-22
PL199298A1 (pl)	1978-03-28
DE2630060C2 (de)	1984-04-19
BE856395A (fr)	1978-01-02
PH14572A (en)	1981-09-24
PT66756A (de)	1977-08-01
JPS535164A (en)	1978-01-18
JPS6026108B2 (ja)	1985-06-21
AU2662077A (en)	1979-01-04
CS204005B2 (en)	1981-03-31
SE431871B (sv)	1984-03-05
ES466852A1 (es)	1978-10-01
PL102918B1 (pl)	1979-05-31
SU680644A3 (ru)	1979-08-15
MX4841E (es)	1982-10-28
IE45109L (en)	1978-01-03
ZA773979B (en)	1979-03-28
DE2630060A1 (de)	1978-01-12
NZ184539A (en)	1980-03-05
DK296477A (da)	1978-01-04
FI771972A (no)	1978-01-04
LU77679A1 (no)	1978-09-14
ES466850A1 (es)	1978-10-01
AT354436B (de)	1979-01-10
IE45109B1 (en)	1982-06-16
NL930111I2 (nl)	1995-04-03
GB1575147A (en)	1980-09-17
SU665800A3 (ru)	1979-05-30
FI64146B (fi)	1983-06-30
NL188643B (nl)	1992-03-16
DK146281B (da)	1983-08-22
NO145951B (no)	1982-03-22
IL52433A0 (en)	1977-10-31
CH633275A5 (de)	1982-11-30
CA1088550A (en)	1980-10-28
YU161977A (en)	1983-01-21
CH633273A5 (de)	1982-11-30
IL52433A (en)	1980-09-16
BG28049A3 (en)	1980-02-25
AU507260B2 (en)	1980-02-07
NL930111I1 (nl)	1993-10-18
NL7707308A (nl)	1978-01-05
HU180429B (en)	1983-03-28
DK146281C (da)	1984-01-30
ES466851A1 (es)	1978-10-01
FR2356642B1 (fr)	1985-07-19
GR63636B (en)	1979-11-27
SE7707689L (sv)	1978-01-04

Publication	Publication Date	Title
NO147243C (no)	1983-03-02	Analogifremgangsmaate for fremstilling av terapeutisk aktive ftalanderivater
NO151321C (no)	1985-03-20	Analogifremgangsmaate for fremstilling av terapeutisk aktive karbostyrilderivater
NO151463C (no)	1985-04-17	Analogifremgangsmaate for fremstilling av terapeutisk aktive kinazolinderivater
NO151411C (no)	1985-04-10	Analogifremgangsmaate for fremstilling av terapeutisk aktive 1-aryloksy-2-hydroksy-3-alkylenaminopropan-derivater
NO800626L (no)	1980-09-08	Analogifremgangsmaate for fremstilling av farmakologisk aktive polyolderivater
NO148813C (no)	1983-12-21	Analogifremgangsmaate for fremstilling av farmakologisk aktive karbostyrilderivater
NO148453C (no)	1983-10-12	Analogifremgangsmaate for fremstilling av terapeutisk aktive spirohydantoinderivater
NO800881L (no)	1980-09-29	Analogifremgangsmaate for fremstilling av terapeutisk aktive kinolonderivater
NO144848C (no)	1981-11-25	Analogifremgangsmaate til fremstilling av terapeutisk virksomme 4-hydroksyfenylalkanolamin-derivater
NO148777C (no)	1984-01-25	Analogifremgangsmaate for fremstilling av terapeutisk aktive antrakinon-derivater
NO149065C (no)	1984-02-08	Analogifremgangsmaate for fremstilling av terapeutisk aktive benzodiazepinderivater
NO150044C (no)	1984-08-22	Analogifremgangsmaate for fremstilling av terapeutisk aktive tetrazol-derivater
NO145842C (no)	1982-06-09	Analogifremgangsmaate for fremstilling av farmakologisk aktive indolizinderivater
NO145951C (no)	1982-06-30	Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazolinderivater
NO144215C (no)	1981-07-15	Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazolin/derivater
NO149313C (no)	1984-03-28	Analogifremgangsmaate for fremstilling av terapeutisk aktive pyridobenzodiazepiner
NO149037C (no)	1984-02-01	Analogifremgangsmaate for fremstilling av terapeutisk aktive pyridobenzodiazepiner
NO148291C (no)	1983-09-14	Analogifremgangsmaate til fremstilling av terapeutisk aktive basisk substituerte teofyllinderivater
NO148454C (no)	1983-10-12	Analogifremgangsmaate for fremstilling av terapeutisk aktive tiazolidin-dionderivater
NO148488C (no)	1983-10-19	Analogifremgangsmaate til fremstilling av terapeutisk aktive acyl-benzimidazol-2-derivater
NO145163C (no)	1982-01-27	Analogifremgangsmaate til fremstilling av terapeutisk aktive antitumorglykosider
NO152172C (no)	1985-08-14	Analogifremgangsmaate for fremstilling av terapeutisk aktive spiro-kinolyl-hydantoin-derivater
NO143903C (no)	1981-05-06	Analogifremgangsmaate for fremstilling av terapeutisk aktive 5-fluorpyrimidin-4-on-derivater
NO146710C (no)	1982-11-24	Analogifremgangsmaate for fremstilling av terapeutisk aktive fenylpiperazinderivater
NO147273C (no)	1983-03-09	Analogifremgangsmaate til fremstilling av terapeutisk aktive cykloheksadien-derivater