MXPA01007963A - Derivados de evermectin. - Google Patents

Derivados de evermectin.

Info

Publication number
MXPA01007963A
MXPA01007963A MXPA01007963A MXPA01007963A MXPA01007963A MX PA01007963 A MXPA01007963 A MX PA01007963A MX PA01007963 A MXPA01007963 A MX PA01007963A MX PA01007963 A MXPA01007963 A MX PA01007963A MX PA01007963 A MXPA01007963 A MX PA01007963A
Authority
MX
Mexico
Prior art keywords
line
carbon atom
avermectin derivatives
double bond
avermectin
Prior art date
Application number
MXPA01007963A
Other languages
English (en)
Inventor
Andreas Turberg
Original Assignee
Kitasato Inst
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kitasato Inst filed Critical Kitasato Inst
Publication of MXPA01007963A publication Critical patent/MXPA01007963A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
MXPA01007963A 1999-02-09 2000-02-09 Derivados de evermectin. MXPA01007963A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3105899 1999-02-09
JP24863399 1999-09-02
PCT/JP2000/000691 WO2000047597A1 (fr) 1999-02-09 2000-02-09 Derives de l'avermectine

Publications (1)

Publication Number Publication Date
MXPA01007963A true MXPA01007963A (es) 2004-01-29

Family

ID=26369507

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA01007963A MXPA01007963A (es) 1999-02-09 2000-02-09 Derivados de evermectin.

Country Status (14)

Country Link
US (1) US6605595B1 (es)
EP (2) EP1160252B1 (es)
JP (1) JP4832645B2 (es)
KR (1) KR20010101819A (es)
CN (2) CN1637011A (es)
AT (1) ATE556083T1 (es)
AU (1) AU769612B2 (es)
BR (1) BR0009861A (es)
CA (1) CA2362253C (es)
ES (1) ES2387384T3 (es)
HK (1) HK1040083A1 (es)
MX (1) MXPA01007963A (es)
NZ (1) NZ514026A (es)
WO (1) WO2000047597A1 (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2001277712A1 (en) * 2000-08-09 2002-02-18 The Kitasato Institute Avermectin derivatives
CA2418975C (en) * 2000-08-09 2012-01-17 Satoshi Omura Avermectin derivatives
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
AR036486A1 (es) * 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
RU2004115744A (ru) * 2001-10-25 2005-04-10 Санкио Лайфтек Компани, Лимитед (Jp) Антигельминтная композиция
TW200407330A (en) 2002-05-07 2004-05-16 Syngenta Participations Ag 4"-Deoxy-4"-(S)-amido avermectin derivatives
GB0302309D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302310D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302547D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
US7396819B2 (en) * 2003-08-08 2008-07-08 Virbac Corporation Anthelmintic formulations
GB0320176D0 (en) * 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
US7582612B2 (en) * 2004-03-12 2009-09-01 Hartz Mountain Corporation Multi-action anthelmintic formulations
CN103360444B (zh) 2012-04-03 2016-05-11 浙江海正药业股份有限公司 抗寄生虫药赛拉菌素的合成新工艺
CN104231022B (zh) * 2013-06-14 2018-10-09 南开大学 一种大环内酯类化合物的制备及应用
CN103421065B (zh) * 2013-07-03 2016-05-18 大庆志飞生物化工有限公司 一类新型阿维菌素衍生物及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4427663A (en) 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4833168A (en) * 1986-10-03 1989-05-23 Merck & Co., Inc. Avermectin reformatsky adducts
US4895837A (en) 1988-01-29 1990-01-23 Merck & Co., Inc. Avermectin derivatives
US4906619A (en) * 1988-07-22 1990-03-06 Merck & Co., Inc. Alkyl avermectin derivatives
US5030622A (en) * 1989-06-02 1991-07-09 Merck & Co., Inc. Avermectin derivatives
JPH0325467A (ja) 1989-06-22 1991-02-04 Konica Corp カラー画像形成装置
JP2888586B2 (ja) 1990-03-05 1999-05-10 社団法人北里研究所 エバーメクチンの特定成分を選択生産するための微生物およびその選択的製造法
JPH0633273A (ja) 1992-07-16 1994-02-08 Asahi Chem Ind Co Ltd Ａｌｃの埋込金属部材用の防錆剤
GB9312154D0 (en) 1993-06-12 1993-07-28 Pfizer Ltd Antiparasitic agents

Also Published As

Publication number Publication date
EP1160252A4 (en) 2002-07-17
CA2362253A1 (en) 2000-08-17
EP1160252B1 (en) 2012-05-02
CN1202116C (zh) 2005-05-18
AU769612B2 (en) 2004-01-29
US6605595B1 (en) 2003-08-12
BR0009861A (pt) 2002-01-15
EP2332949A1 (en) 2011-06-15
JP4832645B2 (ja) 2011-12-07
HK1040083A1 (zh) 2002-05-24
ATE556083T1 (de) 2012-05-15
CN1637011A (zh) 2005-07-13
ES2387384T3 (es) 2012-09-21
WO2000047597A1 (fr) 2000-08-17
NZ514026A (en) 2001-09-28
CA2362253C (en) 2008-09-23
KR20010101819A (ko) 2001-11-14
CN1346362A (zh) 2002-04-24
AU2459000A (en) 2000-08-29
EP1160252A1 (en) 2001-12-05

Similar Documents

Publication Publication Date Title
HK1040083A1 (zh) 愛弗美思汀(avermectin)衍生物
CA2096969A1 (en) 6-0-methylerythromycin a derivatives
HUP0204034A3 (en) Stable salts of novel derivatives of 3,3-diphenylpropylamines
YU74500A (sh) Novi derivat 3-aril-2-hidroksipropionske kiseline (i)
DE69840645D1 (en) Benzamidinderivate
IL145633A0 (en) Pharmaceutical compounds
EP1029860A4 (en) BENZOFURAN DERIVATIVES
AU7948900A (en) 4-oxoquinolizine antimicrobials having 2-pyridone skeletons as the partial structure
EP0241901A3 (en) Cephalosporin derivatives, processes for their preparation and antibacterial agents
BG104447A (en) Biphenylamidine derivatives
HU9502270D0 (en) Novel pyrrolocarbazoles
NZ243695A (en) Iodinated ethers and their preparation
HK1015766A1 (en) 1-methylcarbapenem derivatives
EP1043311A4 (en) BIPHENYLAMIDINE DERIVATIVES
NO990914L (no) Amorfe benzotiofener, fremgangsmÕter for fremstilling og fremgangsmÕter for anvendelse
EP1026162A4 (en) ANTI-RHUMATISMAL AGENT
IL157440A0 (en) Triazole derivatives and pharmaceutical compositions containing the same
EP1074545A4 (en) ISOCHINOLINE SULPHONAMIDE DERIVATIVES AND MEDICINES CONTAINING IT AS AN ACTIVE INGREDIENT
AU1639197A (en) Pyridine derivative, anti-ulcer drug, and antibacterial drug
EP0759297A4 (en) MEDICINE AGAINST PULMONAL HEART PROBLEMS
WO2003034978A3 (en) Antidiabetic 2-substituted-5'-o- (1-boranotriphosphate) adenosine derivatives
IL152632A0 (en) Trimethyldecenyl compounds
DE69620128D1 (de) Herboxidien-Derivate und ihre Herstellung aus einer Streptomyces GEX1 Kultur
EP0376114A3 (en) 9-dihydro-9-0-alkyldesmycosin derivatives
BG102578A (en) 1,3-oxazin-4-on derivatives as herbicides

Legal Events

Date Code Title Description
FG Grant or registration