MA26732A1 - NOVEL PHARMACEUTICAL COMPOSITION COMPRISING AN OUR INHIBITOR, AND METHOD FOR THE PREPARATION THEREOF - Google Patents

NOVEL PHARMACEUTICAL COMPOSITION COMPRISING AN OUR INHIBITOR, AND METHOD FOR THE PREPARATION THEREOF

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Publication number
MA26732A1
MA26732A1 MA25976A MA25976A MA26732A1 MA 26732 A1 MA26732 A1 MA 26732A1 MA 25976 A MA25976 A MA 25976A MA 25976 A MA25976 A MA 25976A MA 26732 A1 MA26732 A1 MA 26732A1
Authority
MA
Morocco
Prior art keywords
preparation
inhibitor
pharmaceutical composition
novel pharmaceutical
treatment
Prior art date
Application number
MA25976A
Other languages
French (fr)
Inventor
David Saltarelli Mario
Adams Lowe John Iii
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of MA26732A1 publication Critical patent/MA26732A1/en

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/13—Amines
    • A61K31/15—Oximes (>C=N—O—); Hydrazines (>N—N<); Hydrazones (>N—N=) ; Imines (C—N=C)
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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Anesthesiology (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

L'INVENTION CONCERNE DES COMPOSITIONS PHARMACEUTIQUES COMPRENANT UN COMPOSÉ INHIBITEUR DE NOS, SEUL OU EN ASSOCIATION AVEC UN ANTAGONISTE DES RÉCEPTEURS DE NK-1 OU UN SSRI. ELLE CONCERNE ÉGALEMENT UN PROCÉDÉ POUR LEUR PRÉPARATION. - APPLICATION : UTILISATION DE CES COMPOSITIONS POUR LE TRAITEMENT DE DIVERS TROUBLES DONT LE TRAITEMENT PEUT eTRE EFFECTUÉ OU FACILITÉ PAR LA MODOFICATION DES RYTHMES CIRCADIENS.THE INVENTION RELATES TO PHARMACEUTICAL COMPOSITIONS COMPRISING AN OUR INHIBITOR COMPOUND, ALONE OR IN ASSOCIATION WITH AN ANTAGONIST OF NK-1 RECEPTORS OR AN SSRI. IT ALSO CONCERNS A PROCESS FOR THEIR PREPARATION. - APPLICATION: USE OF THESE COMPOSITIONS FOR THE TREATMENT OF VARIOUS DISORDERS OF WHICH THE TREATMENT MAY BE CARRIED OUT OR FACILITATED BY MODIFYING CIRCADIAN RHYTHMS.

MA25976A 1999-05-21 2000-05-17 NOVEL PHARMACEUTICAL COMPOSITION COMPRISING AN OUR INHIBITOR, AND METHOD FOR THE PREPARATION THEREOF MA26732A1 (en)

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DE10001785A1 (en) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma Use of NK-1 receptor antagonists for treatment of restless legs syndrome
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
DOP2002000467A (en) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-AMINO-6 (PHENYL REPLACED IN POSITIONS 2,4,5) -PIRIDINES
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
AU2004249441B2 (en) 2003-06-24 2009-11-12 Neurosearch A/S Novel 8-aza-bicyclo(3.2.1)octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
EP1634598A1 (en) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Use of piperazine derivatives and analogues for the manufacture of a medicament for the prophylaxis and/or treatment of disorders of food ingestion
JP5464709B2 (en) 2007-06-08 2014-04-09 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Piperidine / piperazine derivatives
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine/Piperazine derivatives
RU2470017C2 (en) 2007-06-08 2012-12-20 Янссен Фармацевтика Н.В. Piperidine/piperazine derivatives
AU2008258549B2 (en) 2007-06-08 2013-11-14 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
CA2725933C (en) 2008-06-05 2018-01-16 Janssen Pharmaceutica Nv Drug combinations comprising a dgat inhibitor and a ppar-agonist
EP2404902A1 (en) 2009-03-05 2012-01-11 Shionogi&Co., Ltd. Piperidine and pyrrolidine derivatives having npy y5 receptor antagonism
EP2919788A4 (en) 2012-11-14 2016-05-25 Univ Johns Hopkins Methods and compositions for treating schizophrenia
US20220267269A1 (en) * 2019-06-14 2022-08-25 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (pcsk9)
US12115154B2 (en) 2020-12-16 2024-10-15 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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HUP0301287A2 (en) 2003-08-28
SK16602001A3 (en) 2003-03-04
UY26148A1 (en) 2000-12-29
AR022640A1 (en) 2002-09-04
JP2003523941A (en) 2003-08-12
HRP20010862A2 (en) 2003-06-30
DZ3041A1 (en) 2004-03-27
AP2001002326A0 (en) 2001-12-31
NO20015651D0 (en) 2001-11-20
EA200101110A1 (en) 2002-08-29
WO2000071107A8 (en) 2002-01-24
GT200000071A (en) 2001-11-08
WO2000071107A2 (en) 2000-11-30
CN1617743A (en) 2005-05-18
NO20015651L (en) 2002-01-18
EE200100611A (en) 2003-02-17
ZA200109555B (en) 2004-04-07
AU2935300A (en) 2000-12-12
OA11943A (en) 2006-04-12
CA2374668A1 (en) 2000-11-30
TNSN00106A1 (en) 2005-11-10
TR200103351T2 (en) 2002-06-21
PE20010157A1 (en) 2001-02-16
IS6126A (en) 2001-10-26
BG106208A (en) 2002-09-30
PA8494601A1 (en) 2002-08-29
BR0010820A (en) 2002-03-05
MXPA01011978A (en) 2002-05-06
IL145955A0 (en) 2002-07-25
PL358538A1 (en) 2004-08-09
HN2000000045A (en) 2001-03-02
CO5160295A1 (en) 2002-05-30
KR20020010916A (en) 2002-02-06
EP1178784A1 (en) 2002-02-13
HUP0301287A3 (en) 2005-03-29

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