JPS5735561A - Novel alpha- mercaptomethyl acrylic acid derivative - Google Patents
Novel alpha- mercaptomethyl acrylic acid derivativeInfo
- Publication number
- JPS5735561A JPS5735561A JP11212380A JP11212380A JPS5735561A JP S5735561 A JPS5735561 A JP S5735561A JP 11212380 A JP11212380 A JP 11212380A JP 11212380 A JP11212380 A JP 11212380A JP S5735561 A JPS5735561 A JP S5735561A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound shown
- acrylic acid
- mercaptomethyl
- synthesizing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
NEW MATERIAL:An α-(mercaptomethyl)acrylic acid derivative shown by the formula I [R1 is H, lower alkanoyl, (substituted)benzoyl, group shown by the formula II, etc.; R2 is H or lower alkyl].
EXAMPLE: α-(Benzoylthiomethyl)acrylic acid.
USE: A raw material for synthesizing a compound shown by the formula III useful as a hypotensive and an intermediate for synthesizing a drug.
PROCESS: A compound shown by the formula IV (X is Cl, Br, I, methanesulfonyl, or p-toluenesulfonyl) is reacted with a compound shown by the formual R1SH to give the titled compound shown by the formula I. The reaction is carried out in a solvent, e.g., methylene chloride, etc. at -50W100°C, preferably at -10W50°C. The compound shown by the formula I is subjected to catalytic asymmetric hydrogenation in the presence of a rhodium complex containing an optically active phosphine ligand, to give a compound shown by the formula V, a raw material for synthesizing a compound shown by the formula III at one try.
COPYRIGHT: (C)1982,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP11212380A JPS5735561A (en) | 1980-08-13 | 1980-08-13 | Novel alpha- mercaptomethyl acrylic acid derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP11212380A JPS5735561A (en) | 1980-08-13 | 1980-08-13 | Novel alpha- mercaptomethyl acrylic acid derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS5735561A true JPS5735561A (en) | 1982-02-26 |
Family
ID=14578761
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP11212380A Pending JPS5735561A (en) | 1980-08-13 | 1980-08-13 | Novel alpha- mercaptomethyl acrylic acid derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5735561A (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4671928A (en) * | 1984-04-26 | 1987-06-09 | International Business Machines Corporation | Method of controlling the sintering of metal particles |
JPH04356510A (en) * | 1990-06-27 | 1992-12-10 | Elf Atochem Sa | New acrylic compound containing sulfur, its manufacture, and its use in the synthesis of new polymer |
-
1980
- 1980-08-13 JP JP11212380A patent/JPS5735561A/en active Pending
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4671928A (en) * | 1984-04-26 | 1987-06-09 | International Business Machines Corporation | Method of controlling the sintering of metal particles |
JPH04356510A (en) * | 1990-06-27 | 1992-12-10 | Elf Atochem Sa | New acrylic compound containing sulfur, its manufacture, and its use in the synthesis of new polymer |
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