JPS5540616A - Preparation of benzo-hetero-compound - Google Patents
Preparation of benzo-hetero-compoundInfo
- Publication number
- JPS5540616A JPS5540616A JP11310478A JP11310478A JPS5540616A JP S5540616 A JPS5540616 A JP S5540616A JP 11310478 A JP11310478 A JP 11310478A JP 11310478 A JP11310478 A JP 11310478A JP S5540616 A JPS5540616 A JP S5540616A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- benzo
- hetero
- alkoxy
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Quinoline Compounds (AREA)
- Indole Compounds (AREA)
Abstract
PURPOSE: To prepare the title compound useful as an intermeidate of antibiotic agent, by reducing a 4-dihydrocarbostyril derivative which is a known or an easily synthesizable compound.
CONSTITUTION: A benzo-hetero-compound of formulaII(R1 is H, OH, amino, halogen, alkoxy, alkyl, alkanesulfonyloxy or allenesulfonyloxy; R2 is H, halogen, alkoxy, alkyl, or phenylalkoxy; R3 is H, halogen or alkoxy; l is 1W3), e.g. 5- methanesulfonyl-oxy-1,2,3,4-tetrahydroquinoline, is prepared by reducing a 3,4- dihydrocarbostyril derivative of formulaI, e.g. 5-methanesulfonyloxy-3,4-dihydrocarbostyril, preferably with a hydrogenating agent such as sodium borohydride.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP11310478A JPS5540616A (en) | 1978-09-14 | 1978-09-14 | Preparation of benzo-hetero-compound |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP11310478A JPS5540616A (en) | 1978-09-14 | 1978-09-14 | Preparation of benzo-hetero-compound |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5540616A true JPS5540616A (en) | 1980-03-22 |
JPS6237628B2 JPS6237628B2 (en) | 1987-08-13 |
Family
ID=14603577
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP11310478A Granted JPS5540616A (en) | 1978-09-14 | 1978-09-14 | Preparation of benzo-hetero-compound |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5540616A (en) |
Cited By (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4416884A (en) * | 1978-04-12 | 1983-11-22 | Otsuka Pharmaceutical Co., Ltd. | Piperazinylbenzoheterocyclic compounds |
US4552879A (en) * | 1980-11-10 | 1985-11-12 | Otsuka Pharmaceutical Co., Ltd. | Benzoheterocyclic compounds and pharmaceutical composition thereof |
US4594347A (en) * | 1983-01-26 | 1986-06-10 | Otsuka Pharmaceutical Co. Limited | Pyrrolo [3,2,1-ij]-quinoline carboxylic acid compound |
JPS61194074A (en) * | 1985-02-22 | 1986-08-28 | Sumitomo Chem Co Ltd | 7-amino-1-alkyl-6-fluoroquinolin-2(1h)-one and its preparation |
US5283336A (en) * | 1992-09-08 | 1994-02-01 | The United States Of America As Represented By The United States Department Of Energy | Method for preparation of 7-hydroxy-1,2,3,4-tetrahydroquinoline from 1,2,3,4-tetrahydroquinoline |
WO2002006228A1 (en) * | 2000-07-19 | 2002-01-24 | Ube Industries, Ltd. | Process for producing 5-fluorooxyindole and for producing intermediate therefor |
DE102008022221A1 (en) | 2008-05-06 | 2009-11-12 | Universität des Saarlandes | Inhibitors of human aldosterone synthase CYP11B2 |
US8541404B2 (en) | 2009-11-09 | 2013-09-24 | Elexopharm Gmbh | Inhibitors of the human aldosterone synthase CYP11B2 |
US10870721B2 (en) | 2013-06-18 | 2020-12-22 | Panasonic Intellectual Property Management Co., Ltd. | Polyphenylene ether resin composition, prepreg, metal-clad laminate and printed wiring board |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH0519662U (en) * | 1991-05-28 | 1993-03-12 | 株式会社中村自工 | Drive shaft |
Citations (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS4876898A (en) * | 1971-12-30 | 1973-10-16 | ||
JPS4941539A (en) * | 1972-05-17 | 1974-04-18 | ||
JPS4982672A (en) * | 1972-12-21 | 1974-08-08 | ||
JPS4982670A (en) * | 1972-12-18 | 1974-08-08 | ||
JPS49125530A (en) * | 1973-03-26 | 1974-12-02 | ||
JPS5024296A (en) * | 1973-04-05 | 1975-03-15 | ||
JPS50108271A (en) * | 1974-02-09 | 1975-08-26 | ||
JPS50108277A (en) * | 1974-02-12 | 1975-08-26 | ||
US3917609A (en) * | 1973-06-27 | 1975-11-04 | Minnesota Mining & Mfg | Pyrroloquinoline carboxylic acids and derivatives |
JPS51146476A (en) * | 1975-06-06 | 1976-12-16 | Chinoin Gyogyszer Es Vegyeszet | New preparation method of quinolinee33carbonic acid |
JPS5236606A (en) * | 1975-09-12 | 1977-03-22 | Tanabe Seiyaku Co Ltd | Process for preparation of amino compounds |
JPS5365887A (en) * | 1976-11-22 | 1978-06-12 | Kyorin Seiyaku Kk | Substituted quinoline*arboxylate and process for preparing same |
JPS5382799A (en) * | 1976-12-28 | 1978-07-21 | Kyorin Seiyaku Kk | Substituted pyroloquinolinecarboxylate and process for preparing same |
-
1978
- 1978-09-14 JP JP11310478A patent/JPS5540616A/en active Granted
Patent Citations (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS4876898A (en) * | 1971-12-30 | 1973-10-16 | ||
JPS4941539A (en) * | 1972-05-17 | 1974-04-18 | ||
JPS4982670A (en) * | 1972-12-18 | 1974-08-08 | ||
JPS4982672A (en) * | 1972-12-21 | 1974-08-08 | ||
JPS49125530A (en) * | 1973-03-26 | 1974-12-02 | ||
JPS5024296A (en) * | 1973-04-05 | 1975-03-15 | ||
US3917609A (en) * | 1973-06-27 | 1975-11-04 | Minnesota Mining & Mfg | Pyrroloquinoline carboxylic acids and derivatives |
JPS50108271A (en) * | 1974-02-09 | 1975-08-26 | ||
JPS50108277A (en) * | 1974-02-12 | 1975-08-26 | ||
JPS51146476A (en) * | 1975-06-06 | 1976-12-16 | Chinoin Gyogyszer Es Vegyeszet | New preparation method of quinolinee33carbonic acid |
JPS5236606A (en) * | 1975-09-12 | 1977-03-22 | Tanabe Seiyaku Co Ltd | Process for preparation of amino compounds |
JPS5365887A (en) * | 1976-11-22 | 1978-06-12 | Kyorin Seiyaku Kk | Substituted quinoline*arboxylate and process for preparing same |
JPS5382799A (en) * | 1976-12-28 | 1978-07-21 | Kyorin Seiyaku Kk | Substituted pyroloquinolinecarboxylate and process for preparing same |
Cited By (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4416884A (en) * | 1978-04-12 | 1983-11-22 | Otsuka Pharmaceutical Co., Ltd. | Piperazinylbenzoheterocyclic compounds |
US4552879A (en) * | 1980-11-10 | 1985-11-12 | Otsuka Pharmaceutical Co., Ltd. | Benzoheterocyclic compounds and pharmaceutical composition thereof |
US4594347A (en) * | 1983-01-26 | 1986-06-10 | Otsuka Pharmaceutical Co. Limited | Pyrrolo [3,2,1-ij]-quinoline carboxylic acid compound |
JPS61194074A (en) * | 1985-02-22 | 1986-08-28 | Sumitomo Chem Co Ltd | 7-amino-1-alkyl-6-fluoroquinolin-2(1h)-one and its preparation |
US5283336A (en) * | 1992-09-08 | 1994-02-01 | The United States Of America As Represented By The United States Department Of Energy | Method for preparation of 7-hydroxy-1,2,3,4-tetrahydroquinoline from 1,2,3,4-tetrahydroquinoline |
WO2002006228A1 (en) * | 2000-07-19 | 2002-01-24 | Ube Industries, Ltd. | Process for producing 5-fluorooxyindole and for producing intermediate therefor |
US6900335B2 (en) | 2000-07-19 | 2005-05-31 | Ube Industries, Ltd. | Process for producing 5-fluorooxindole and for producing intermediates therefor |
US7342040B2 (en) | 2000-07-19 | 2008-03-11 | Ube Industries, Ltd. | 5-fluorooxindole-3-carboxylic acid ester |
DE102008022221A1 (en) | 2008-05-06 | 2009-11-12 | Universität des Saarlandes | Inhibitors of human aldosterone synthase CYP11B2 |
US8685960B2 (en) | 2008-05-06 | 2014-04-01 | Elexopharm Gmbh | 6-pyridin-3-yl-3,4-dihydro-1h-quinolin-2-one derivatives and related compounds as inhibitors of the human aldosterone synthase CYP11B2 |
US8541404B2 (en) | 2009-11-09 | 2013-09-24 | Elexopharm Gmbh | Inhibitors of the human aldosterone synthase CYP11B2 |
US10870721B2 (en) | 2013-06-18 | 2020-12-22 | Panasonic Intellectual Property Management Co., Ltd. | Polyphenylene ether resin composition, prepreg, metal-clad laminate and printed wiring board |
Also Published As
Publication number | Publication date |
---|---|
JPS6237628B2 (en) | 1987-08-13 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
JPS5540616A (en) | Preparation of benzo-hetero-compound | |
DE3264760D1 (en) | New pyrazoline derivatives, method of preparing the new compounds, as well as insecticidal compositions on the basis of these compounds | |
JPS5212109A (en) | Process for preparation of alkylglycerylether | |
JPS5692239A (en) | Preparation of 5-oxohexyl compound | |
JPS53111096A (en) | 1-azaxanthone-3-carboxylic acid derivative and its preparation | |
JPS5424829A (en) | Organic phosphate compound, its preparation, and insecticide, miticide and nematocide containing the same | |
JPS5742643A (en) | 6,10,14,18-tetramethyl-5,9,13,17-nonadecatetraene-2-ol | |
JPS53132547A (en) | Novel trisazo compound and its preparation | |
ES485157A1 (en) | Benzimidazolyl-2-carbamic acid esters, medicaments based thereon and process for their preparation. | |
JPS53101308A (en) | Derivative of 5,6-dihydro-2h-pyran and its preparation | |
AU8714082A (en) | N-substituted-tetrahydroisophthalimide derivatives | |
JPS5414951A (en) | Preparation of vitamin d derivatives | |
JPS51122043A (en) | Process for preparation of 3-hydroxy-5- cycloxycyclopento-1-ene deriva tives | |
JPS6485970A (en) | Saccharoascorbic acid ester and production thereof | |
JPS53103415A (en) | Preparation of trihalocarboxylic acid ester | |
JPS5422376A (en) | Carbostyril derivative | |
JPS5412385A (en) | Carbostyril derivative | |
JPS5368777A (en) | Preparation of phenyathridine | |
JPS5422353A (en) | 2-chloro-2-cyano-7-alkylidene-bicyclo(2,2,1)-5-heptene and its preparation | |
JPS5692229A (en) | Preparation of 5-hexynyl alcohol | |
JPS5412355A (en) | Alkyl cyclohexyldichlorosilane compounds and their preparation | |
JPS53149924A (en) | Beta-hydroxy-alpha-amino acid compound and its preparation | |
JPS5422355A (en) | 7-alkylnorcamphor, its preparation, and perfume composition comprising the compounds | |
JPS53135998A (en) | Preparation of 6 alpha-acylaminopenicillanic acid 1-oxide | |
JPS5422354A (en) | 2-chloro-2-cyano-7-aklylbicyclo-(2.2.1)heptane and its preparation |