FR2357574A1 - Nouveaux derives 16-acylthio de l'acide fusidique, utiles notamment comme antimicrobiens et leur procede de preparation - Google Patents

Nouveaux derives 16-acylthio de l'acide fusidique, utiles notamment comme antimicrobiens et leur procede de preparation

Info

Publication number
FR2357574A1
FR2357574A1 FR7720523A FR7720523A FR2357574A1 FR 2357574 A1 FR2357574 A1 FR 2357574A1 FR 7720523 A FR7720523 A FR 7720523A FR 7720523 A FR7720523 A FR 7720523A FR 2357574 A1 FR2357574 A1 FR 2357574A1
Authority
FR
France
Prior art keywords
antimicrobials
useful
new
preparation process
fusidic acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7720523A
Other languages
English (en)
Other versions
FR2357574B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SARATH
Original Assignee
SARATH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SARATH filed Critical SARATH
Publication of FR2357574A1 publication Critical patent/FR2357574A1/fr
Application granted granted Critical
Publication of FR2357574B1 publication Critical patent/FR2357574B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0027—Azides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/007—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 17 (20)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/003—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring the S atom directly linked to a ring carbon atom of the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

Les médicaments sont des composés de formule générale:
FR7720523A 1976-07-05 1977-07-04 Nouveaux derives 16-acylthio de l'acide fusidique, utiles notamment comme antimicrobiens et leur procede de preparation Granted FR2357574A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB27921/76A GB1581335A (en) 1976-07-05 1976-07-05 16-s-acyl derivatives of fusidic acid

Publications (2)

Publication Number Publication Date
FR2357574A1 true FR2357574A1 (fr) 1978-02-03
FR2357574B1 FR2357574B1 (fr) 1979-07-20

Family

ID=10267438

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7720523A Granted FR2357574A1 (fr) 1976-07-05 1977-07-04 Nouveaux derives 16-acylthio de l'acide fusidique, utiles notamment comme antimicrobiens et leur procede de preparation

Country Status (22)

Country Link
US (1) US4119717A (fr)
JP (1) JPS535152A (fr)
AT (1) AT354625B (fr)
AU (1) AU516152B2 (fr)
BE (1) BE856464A (fr)
CA (1) CA1100941A (fr)
DE (1) DE2730196C2 (fr)
DK (1) DK148390B (fr)
FI (1) FI58136C (fr)
FR (1) FR2357574A1 (fr)
GB (1) GB1581335A (fr)
GR (1) GR63210B (fr)
IE (1) IE45217B1 (fr)
IT (1) IT1083082B (fr)
LU (1) LU77683A1 (fr)
NL (1) NL7707221A (fr)
NZ (1) NZ184408A (fr)
PH (1) PH14058A (fr)
PT (1) PT66759B (fr)
SE (1) SE436752B (fr)
YU (1) YU165477A (fr)
ZA (1) ZA773739B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4162259A (en) * 1975-12-03 1979-07-24 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske fabrik Produktionsaktienselskab) Fusidic acid derivatives
US4548922A (en) * 1983-06-06 1985-10-22 Beth Israel Hospital Drug administration
US4959358A (en) * 1983-06-06 1990-09-25 Beth Israel Hospital Assn. Drug administration
US4746508A (en) * 1983-06-06 1988-05-24 Beth Israel Hospital Assn. Drug administration
US4994439A (en) * 1989-01-19 1991-02-19 California Biotechnology Inc. Transmembrane formulations for drug administration
GB9518883D0 (en) * 1995-09-15 1995-11-15 Leo Pharm Prod Ltd Chemical compounds
MY140194A (en) * 2003-07-16 2009-11-30 Leo Pharma As Novel fusidic acid derivatives
WO2008034796A2 (fr) * 2006-09-19 2008-03-27 Solvay Pharmaceuticals Gmbh Triazoles thérapeutiquement actives et leur utilisation
PT106679B (pt) 2012-11-27 2015-03-25 Hovione Farmaciencia Sa Formulações tópicas de tetraciclinas, sua preparação e usos

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2315296A1 (fr) * 1975-06-25 1977-01-21 Sarath Nouveaux 16-ethers de derives d'acide fusidique, utiles notamment comme antimicrobiens, et leur procede de preparation

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1490852A (en) * 1974-09-12 1977-11-02 Leo Pharm Prod Ltd Fusidic acid derivatives
US4060606A (en) * 1975-06-25 1977-11-29 Leo Pharmaceutical Products Ltd. A/S 16-Ethers of fusidic acid derivatives

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2315296A1 (fr) * 1975-06-25 1977-01-21 Sarath Nouveaux 16-ethers de derives d'acide fusidique, utiles notamment comme antimicrobiens, et leur procede de preparation

Also Published As

Publication number Publication date
PH14058A (en) 1980-12-29
FR2357574B1 (fr) 1979-07-20
YU165477A (en) 1982-06-30
ATA455777A (de) 1979-06-15
LU77683A1 (fr) 1978-01-31
PT66759A (en) 1977-08-01
AT354625B (de) 1979-01-25
SE7707749L (sv) 1978-01-06
FI58136C (fi) 1980-12-10
IT1083082B (it) 1985-05-21
NL7707221A (nl) 1978-01-09
BE856464A (fr) 1978-01-04
PT66759B (en) 1978-12-14
AU2643877A (en) 1979-01-04
NZ184408A (en) 1980-04-28
JPS6238360B2 (fr) 1987-08-17
ZA773739B (en) 1978-05-30
GB1581335A (en) 1980-12-10
GR63210B (en) 1979-10-08
FI58136B (fi) 1980-08-29
IE45217L (en) 1978-01-05
JPS535152A (en) 1978-01-18
FI772066A (fr) 1978-01-06
AU516152B2 (en) 1981-05-21
DE2730196A1 (de) 1978-01-19
DK294177A (da) 1978-01-06
CA1100941A (fr) 1981-05-12
SE436752B (sv) 1985-01-21
DE2730196C2 (de) 1987-03-05
DK148390B (da) 1985-06-24
US4119717A (en) 1978-10-10
IE45217B1 (en) 1982-07-14

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Legal Events

Date Code Title Description
TP Transmission of property
ST Notification of lapse