FI973207A - Heterosyklisiä yhdisteitä - Google Patents

Heterosyklisiä yhdisteitä Download PDF

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Publication number
FI973207A
FI973207A FI973207A FI973207A FI973207A FI 973207 A FI973207 A FI 973207A FI 973207 A FI973207 A FI 973207A FI 973207 A FI973207 A FI 973207A FI 973207 A FI973207 A FI 973207A
Authority
FI
Finland
Prior art keywords
heterocyclic compounds
chem
halogen atom
formula
halogenocyclopropyl
Prior art date
Application number
FI973207A
Other languages
English (en)
Swedish (sv)
Other versions
FI973207A0 (fi
Inventor
Makoto Takemura
Youichi Kimura
Katsuhiro Kawakami
Kenichi Kimura
Hitoshi Ohki
Norikazu Matsuhashi
Haruko Kawato
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Publication of FI973207A0 publication Critical patent/FI973207A0/fi
Publication of FI973207A publication Critical patent/FI973207A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Use Of Switch Circuits For Exchanges And Methods Of Control Of Multiplex Exchanges (AREA)
  • Earth Drilling (AREA)
  • Stereophonic System (AREA)
FI973207A 1995-02-02 1997-08-01 Heterosyklisiä yhdisteitä FI973207A (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP1561495 1995-02-02
JP1948195 1995-02-07
JP1947895 1995-02-07
PCT/JP1996/000208 WO1996023782A1 (fr) 1995-02-02 1996-02-01 Composes heterocycliques

Publications (2)

Publication Number Publication Date
FI973207A0 FI973207A0 (fi) 1997-08-01
FI973207A true FI973207A (fi) 1997-10-01

Family

ID=27281082

Family Applications (1)

Application Number Title Priority Date Filing Date
FI973207A FI973207A (fi) 1995-02-02 1997-08-01 Heterosyklisiä yhdisteitä

Country Status (13)

Country Link
US (1) US5849757A (fi)
EP (2) EP1304329B1 (fi)
KR (1) KR100389773B1 (fi)
AT (2) ATE411309T1 (fi)
CA (1) CA2212007C (fi)
DE (2) DE69627985T2 (fi)
DK (1) DK0807630T3 (fi)
ES (2) ES2315432T3 (fi)
FI (1) FI973207A (fi)
NO (1) NO314546B1 (fi)
PT (1) PT807630E (fi)
TW (1) TW487701B (fi)
WO (1) WO1996023782A1 (fi)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0911328T3 (da) * 1995-11-22 2006-06-06 Daiichi Seiyaku Co Substituerede aminocycloalkylpyrrolidinderivater
US6121285A (en) 1995-11-22 2000-09-19 Daiichi Pharmaceutical Co., Ltd. Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
TW519542B (en) * 1996-09-27 2003-02-01 Daiichi Seiyaku Co Bicyclic amine derivative
ZA984527B (en) * 1997-05-30 1998-12-03 Daiichi Seiyaku Co Substituted cyclobutylamine derivative
AR013493A1 (es) 1997-09-15 2000-12-27 Procter & Gamble COMPUESTO DE QUINOLONA, SU USO PARA LA FABRICACIoN DE UN MEDICAMENTO Y COMPOSICIoN FARMACEUTICA QUE LO COMPRENDE
GB9822440D0 (en) * 1998-10-14 1998-12-09 Smithkline Beecham Plc Medicaments
WO2000055116A1 (fr) * 1999-03-17 2000-09-21 Daiichi Pharmaceutical Co., Ltd. Procede de production de derives d'acide 5-amino-8- alkylquinolo necarboxylique, et produits intermediaires intervenant dans la production
US6900225B2 (en) * 2000-03-31 2005-05-31 Daiichi Pharmaceutical Co., Ltd. Quinolonecarboxylic acid derivative
AU2405002A (en) * 2000-11-20 2002-05-27 Daiichi Seiyaku Co Dehalogeno compounds
GB0112834D0 (en) * 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
CN100422170C (zh) * 2002-05-17 2008-10-01 第一制药株式会社 喹诺酮羧酸衍生物的制备方法
US6875784B2 (en) 2002-10-09 2005-04-05 Pharmacia & Upjohn Company Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives
US7915418B2 (en) * 2003-06-06 2011-03-29 Daiichi Pharmaceutical Co., Ltd. Intermediates and process for the production of optically active quinolonecarboxylic acid derivatives
JP4616770B2 (ja) * 2003-06-19 2011-01-19 第一三共株式会社 選択的なアミノ置換基導入法
US7723524B2 (en) * 2003-09-29 2010-05-25 Daiichi Pharmaceutical Co., Ltd. 8-cyanoquinolonecarboxylic acid derivative
ES2537976T3 (es) 2003-12-12 2015-06-16 Daiichi Sankyo Company, Limited Compuestos intermedios para la producción de derivados de ciclopropilamina ópticamente activos y procedimiento para la producción de los compuestos intermedios
DK2001862T3 (da) 2006-03-28 2011-08-08 Warner Chilcott Co Llc Malatsalte og polymorfe af (3S,5S)-7-[3-amino-5-methyl-piperidinyl]-1-cyklopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolincarboxylsyre
EP1999125A2 (en) 2006-03-28 2008-12-10 The Procter and Gamble Company A coupling process for preparing quinolone intermediates
BRPI0720771A2 (pt) * 2007-01-05 2014-07-15 Daiichi Sankyo Co Ltd Composto, droga, agentes antibacteriano e terapêutico para infecções, métodos para tratar doenças e infecções e para produzir uma droga, um agente antibacteriano e um agente terapêutico para infecções, e, uso do composto.
US8278313B2 (en) 2008-03-11 2012-10-02 Abbott Laboratories Macrocyclic spiro pyrimidine derivatives
US8436005B2 (en) 2008-04-03 2013-05-07 Abbott Laboratories Macrocyclic pyrimidine derivatives
US10300155B2 (en) 2015-12-31 2019-05-28 Washington University Alpha-synuclein ligands

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5772981A (en) * 1980-10-22 1982-05-07 Dainippon Pharmaceut Co Ltd 1,8-naphthyridine derivative and its salt
CS274601B2 (en) * 1983-07-27 1991-09-15 Dainippon Pharmaceutical Co Method of 1,8-naphthyridine derivative production
JPS60260577A (ja) * 1984-06-06 1985-12-23 Dainippon Pharmaceut Co Ltd 1,8−ナフチリジン誘導体
ATE75740T1 (de) * 1985-06-26 1992-05-15 Daiichi Seiyaku Co Pyridoncarbonsaeurederivate.
JPH0676400B2 (ja) * 1987-08-25 1994-09-28 大日本製薬株式会社 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
IL90062A (en) * 1988-04-27 1994-10-07 Daiichi Seiyaku Co History of pyridonecarboxylic acid, their preparation and pharmaceutical preparations containing them
JP2844079B2 (ja) * 1988-05-23 1999-01-06 塩野義製薬株式会社 ピリドンカルボン酸系抗菌剤
HU219403B (hu) * 1989-08-16 2001-04-28 Pfizer Inc. Azabiciklo-csoporttal helyettesített kinolon- és naftiridon-karbonsavak és eljárás ezek előállítására
KR100232937B1 (ko) * 1991-05-28 1999-12-01 스즈키 다다시 피리돈카복실산 유도체 및 이를 함유하는 항균제
KR960011370B1 (ko) * 1991-12-31 1996-08-22 재단법인 한국화학연구소 스피로알킬아민 유도체와 그의 제조방법
EP0550016A1 (en) * 1991-12-31 1993-07-07 Korea Research Institute Of Chemical Technology Novel quinolone carboxylic acid derivatives and processes for preparing same
US5990106A (en) * 1994-02-04 1999-11-23 Dainippon Pharmaceutical Co., Ltd. Bicyclic amino group-substituted pyridonecarboxylic acid derivatives, esters thereof and salts thereof, and bicyclic amines useful as intermediates thereof
DK0911328T3 (da) * 1995-11-22 2006-06-06 Daiichi Seiyaku Co Substituerede aminocycloalkylpyrrolidinderivater

Also Published As

Publication number Publication date
EP0807630A4 (en) 1998-05-13
EP1304329B1 (en) 2008-10-15
CA2212007A1 (en) 1996-08-08
DK0807630T3 (da) 2003-09-01
EP0807630A1 (en) 1997-11-19
DE69627985D1 (de) 2003-06-12
NO973530D0 (no) 1997-07-31
WO1996023782A1 (fr) 1996-08-08
EP1304329A2 (en) 2003-04-23
ES2315432T3 (es) 2009-04-01
PT807630E (pt) 2003-08-29
US5849757A (en) 1998-12-15
DE69637717D1 (de) 2008-11-27
FI973207A0 (fi) 1997-08-01
NO314546B1 (no) 2003-04-07
TW487701B (en) 2002-05-21
KR19980701860A (ko) 1998-06-25
EP1304329A3 (en) 2004-09-15
CA2212007C (en) 2004-09-14
ES2198474T3 (es) 2004-02-01
KR100389773B1 (ko) 2003-10-23
NO973530L (no) 1997-10-02
EP0807630B1 (en) 2003-05-07
ATE411309T1 (de) 2008-10-15
DE69627985T2 (de) 2004-02-19
ATE239720T1 (de) 2003-05-15

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