DK1664041T3 - Phenylcarboxamidforbindelser, der er egnede til behandling af smerter - Google Patents

Phenylcarboxamidforbindelser, der er egnede til behandling af smerter

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Publication number
DK1664041T3
DK1664041T3 DK04784626T DK04784626T DK1664041T3 DK 1664041 T3 DK1664041 T3 DK 1664041T3 DK 04784626 T DK04784626 T DK 04784626T DK 04784626 T DK04784626 T DK 04784626T DK 1664041 T3 DK1664041 T3 DK 1664041T3
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Prior art keywords
pain
treatment
compounds suitable
phenylene compound
animal
Prior art date
Application number
DK04784626T
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English (en)
Inventor
Qun Sun
Original Assignee
Euro Celtique Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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Publication of DK1664041T3 publication Critical patent/DK1664041T3/da

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/56Amides

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Diabetes (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Psychology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Reproductive Health (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Virology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
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DK04784626T 2003-09-22 2004-09-21 Phenylcarboxamidforbindelser, der er egnede til behandling af smerter DK1664041T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50467903P 2003-09-22 2003-09-22
PCT/US2004/030824 WO2005030766A1 (en) 2003-09-22 2004-09-21 Phenyl - carboxamide compounds useful for treating pain

Publications (1)

Publication Number Publication Date
DK1664041T3 true DK1664041T3 (da) 2008-10-27

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Family Applications (2)

Application Number Title Priority Date Filing Date
DK04784626T DK1664041T3 (da) 2003-09-22 2004-09-21 Phenylcarboxamidforbindelser, der er egnede til behandling af smerter
DK08011788.0T DK2017276T3 (da) 2003-09-22 2004-09-21 Phenylcarboxamid-forbindelser til behandling af smerte

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Application Number Title Priority Date Filing Date
DK08011788.0T DK2017276T3 (da) 2003-09-22 2004-09-21 Phenylcarboxamid-forbindelser til behandling af smerte

Country Status (17)

Country Link
US (3) US7799807B2 (da)
EP (2) EP2017276B1 (da)
JP (2) JP4634385B2 (da)
CN (1) CN1856489A (da)
AT (2) ATE496048T1 (da)
AU (1) AU2004276251B2 (da)
CA (1) CA2537010A1 (da)
CY (2) CY1108367T1 (da)
DE (2) DE602004014791D1 (da)
DK (2) DK1664041T3 (da)
ES (2) ES2309564T3 (da)
HK (1) HK1094191A1 (da)
HR (2) HRP20080492T3 (da)
PL (2) PL1664041T3 (da)
PT (2) PT1664041E (da)
SI (2) SI1664041T1 (da)
WO (1) WO2005030766A1 (da)

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JP4077320B2 (ja) 2001-01-29 2008-04-16 塩野義製薬株式会社 5−メチル−1−フェニル−2−(1h)−ピリドンを有効成分として含有する医薬製剤
US7582635B2 (en) 2002-12-24 2009-09-01 Purdue Pharma, L.P. Therapeutic agents useful for treating pain
DE602004021206D1 (de) * 2003-07-24 2009-07-02 Euro Celtique Sa Zur Behandlung oder Vorbeugung von Schmerzen geeignete Heteroaryl-Tetrahydropiperidyl-Verbindungen
MXPA06003123A (es) * 2003-09-22 2006-05-31 Euro Celtique Sa Agentes terapeuticos utiles para el tratamiento del dolor.
EP2017276B1 (en) 2003-09-22 2011-01-19 Euro-Celtique S.A. Phenyl-carboxamide compounds useful for treating pain
US20050197364A1 (en) 2003-10-07 2005-09-08 Kelly Michael G. Amide compounds as ion channel ligands and uses thereof
ES2531621T3 (es) 2005-07-22 2015-03-18 Mochida Pharmaceutical Co., Ltd. Derivado de heterociclidenacetamida novedoso
US20080051380A1 (en) 2006-08-25 2008-02-28 Auerbach Alan H Methods and compositions for treating cancer
US7645767B2 (en) * 2006-08-31 2010-01-12 Trinity Laboratories, Inc. Pharmaceutical compositions for treating chronic pain and pain associated with neuropathy
PE20081692A1 (es) 2007-01-24 2008-12-18 Mochida Pharm Co Ltd Nuevo derivado de heterocicliden acetamida
US8759362B2 (en) * 2008-10-24 2014-06-24 Purdue Pharma L.P. Bicycloheteroaryl compounds and their use as TRPV1 ligands
US8703962B2 (en) * 2008-10-24 2014-04-22 Purdue Pharma L.P. Monocyclic compounds and their use as TRPV1 ligands
JP2011057661A (ja) * 2009-08-14 2011-03-24 Bayer Cropscience Ag 殺虫性カルボキサミド類
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