DK0633886T3 - Farmaceutisk aktive bicyclisk-heterocycliske aminer - Google Patents

Farmaceutisk aktive bicyclisk-heterocycliske aminer

Info

Publication number
DK0633886T3
DK0633886T3 DK93908303T DK93908303T DK0633886T3 DK 0633886 T3 DK0633886 T3 DK 0633886T3 DK 93908303 T DK93908303 T DK 93908303T DK 93908303 T DK93908303 T DK 93908303T DK 0633886 T3 DK0633886 T3 DK 0633886T3
Authority
DK
Denmark
Prior art keywords
pharmaceutically active
heterocyclic amines
active bicyclic
bicyclic
xxx
Prior art date
Application number
DK93908303T
Other languages
English (en)
Inventor
Gordon L Bundy
Eric Jon Jacobsen
Donald E Ayer
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Application granted granted Critical
Publication of DK0633886T3 publication Critical patent/DK0633886T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK93908303T 1992-04-03 1993-03-16 Farmaceutisk aktive bicyclisk-heterocycliske aminer DK0633886T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86364692A 1992-04-03 1992-04-03
PCT/US1993/002188 WO1993020078A1 (en) 1992-04-03 1993-03-16 Pharmaceutically active bicyclic-heterocyclic amines

Publications (1)

Publication Number Publication Date
DK0633886T3 true DK0633886T3 (da) 2000-12-18

Family

ID=25341481

Family Applications (1)

Application Number Title Priority Date Filing Date
DK93908303T DK0633886T3 (da) 1992-04-03 1993-03-16 Farmaceutisk aktive bicyclisk-heterocycliske aminer

Country Status (21)

Country Link
EP (1) EP0633886B1 (da)
JP (1) JPH08502721A (da)
KR (1) KR100284473B1 (da)
AT (1) ATE197051T1 (da)
AU (1) AU675932B2 (da)
CA (1) CA2130937A1 (da)
CZ (1) CZ236494A3 (da)
DE (1) DE69329574T2 (da)
DK (1) DK0633886T3 (da)
ES (1) ES2150941T3 (da)
FI (1) FI944602A (da)
GR (1) GR3035188T3 (da)
HU (1) HUT70954A (da)
LV (1) LV12794B (da)
MX (1) MX9301847A (da)
NO (1) NO303542B1 (da)
PL (2) PL175327B1 (da)
PT (1) PT633886E (da)
RU (1) RU2103272C1 (da)
SK (1) SK119194A3 (da)
WO (1) WO1993020078A1 (da)

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US6680322B2 (en) 1999-12-02 2004-01-20 Osi Pharmaceuticals, Inc. Compounds specific to adenosine A1 receptors and uses thereof
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US7834014B2 (en) 2003-04-09 2010-11-16 Biogen Idec Ma Inc. A2a adenosine receptor antagonists
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AU2005264998A1 (en) 2004-06-17 2006-01-26 Wyeth The present invention relates to methods of making Gonadotropin Releasing Hormone ('GnRH') (also known as Leutinizing Hormone Releasing Hormone) receptor antagonists
RU2007101705A (ru) 2004-06-18 2008-07-27 Биолипокс Аб (Se) Индолы, полезные для лечения воспаления
FR2880626B1 (fr) * 2005-01-13 2008-04-18 Aventis Pharma Sa Derives de la purine, compositions les contenant et utilisation
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US7531542B2 (en) 2005-05-18 2009-05-12 Wyeth Benzooxazole and benzothiazole antagonists of gonadotropin releasing hormone receptor
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KR20110098908A (ko) * 2008-11-11 2011-09-02 엑스커버리 홀딩 컴퍼니 엘엘씨 ＰＩ3Ｋ/ｍＴＯＲ 키나제 억제제
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GB864145A (en) * 1959-06-02 1961-03-29 Thomae Gmbh Dr K Novel purines and a process for their manufacture
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Also Published As

Publication number Publication date
WO1993020078A1 (en) 1993-10-14
AU675932B2 (en) 1997-02-27
PL175347B1 (pl) 1998-12-31
MX9301847A (es) 1993-10-01
NO943655D0 (no) 1994-09-30
DE69329574D1 (de) 2000-11-23
DE69329574T2 (de) 2001-05-31
EP0633886B1 (en) 2000-10-18
FI944602A0 (fi) 1994-10-03
CZ236494A3 (en) 1994-12-15
ES2150941T3 (es) 2000-12-16
EP0633886A1 (en) 1995-01-18
NO303542B1 (no) 1998-07-27
KR100284473B1 (ko) 2001-04-02
PL175327B1 (pl) 1998-12-31
LV12794B (en) 2002-06-20
KR950700912A (ko) 1995-02-20
RU2103272C1 (ru) 1998-01-27
CA2130937A1 (en) 1993-10-14
GR3035188T3 (en) 2001-04-30
NO943655L (no) 1994-12-05
SK119194A3 (en) 1995-05-10
HU9402829D0 (en) 1995-02-28
AU3917493A (en) 1993-11-08
PT633886E (pt) 2001-03-30
FI944602A (fi) 1994-10-03
HUT70954A (en) 1995-11-28
JPH08502721A (ja) 1996-03-26
LV12794A (en) 2002-02-20
ATE197051T1 (de) 2000-11-15
RU94042466A (ru) 1996-07-20

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