BR9709974A - Derivados de 2-(2-oxo-etidileno)-imidazolidin-4-ona e seu uso como inibidores da transferase da proteina de farnesila - Google Patents

Derivados de 2-(2-oxo-etidileno)-imidazolidin-4-ona e seu uso como inibidores da transferase da proteina de farnesila

Info

Publication number
BR9709974A
BR9709974A BR9709974A BR9709974A BR9709974A BR 9709974 A BR9709974 A BR 9709974A BR 9709974 A BR9709974 A BR 9709974A BR 9709974 A BR9709974 A BR 9709974A BR 9709974 A BR9709974 A BR 9709974A
Authority
BR
Brazil
Prior art keywords
ethidylene
imidazolidin
oxo
derivatives
protein transferase
Prior art date
Application number
BR9709974A
Other languages
English (en)
Inventor
Joseph Peter Henry
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of BR9709974A publication Critical patent/BR9709974A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BR9709974A 1996-06-27 1997-05-22 Derivados de 2-(2-oxo-etidileno)-imidazolidin-4-ona e seu uso como inibidores da transferase da proteina de farnesila BR9709974A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2069696P 1996-06-27 1996-06-27
PCT/IB1997/000584 WO1997049700A1 (en) 1996-06-27 1997-05-22 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one and their use as farnesyl protein transferase inhibitors

Publications (1)

Publication Number Publication Date
BR9709974A true BR9709974A (pt) 1999-08-10

Family

ID=21800047

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9709974A BR9709974A (pt) 1996-06-27 1997-05-22 Derivados de 2-(2-oxo-etidileno)-imidazolidin-4-ona e seu uso como inibidores da transferase da proteina de farnesila

Country Status (13)

Country Link
US (1) US6071935A (pt)
EP (1) EP0907649A1 (pt)
JP (1) JPH11512750A (pt)
AP (1) AP9701039A0 (pt)
AU (1) AU2710597A (pt)
BR (1) BR9709974A (pt)
CA (1) CA2259222A1 (pt)
GT (1) GT199700074A (pt)
ID (1) ID17053A (pt)
MA (1) MA26432A1 (pt)
TN (1) TNSN97110A1 (pt)
WO (1) WO1997049700A1 (pt)
ZA (1) ZA975675B (pt)

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Also Published As

Publication number Publication date
WO1997049700A1 (en) 1997-12-31
ZA975675B (en) 1998-01-28
US6071935A (en) 2000-06-06
TNSN97110A1 (fr) 2005-03-15
EP0907649A1 (en) 1999-04-14
AU2710597A (en) 1998-01-14
ID17053A (id) 1997-12-04
AP9701039A0 (en) 1997-07-31
JPH11512750A (ja) 1999-11-02
CA2259222A1 (en) 1997-12-31
MA26432A1 (fr) 2004-12-20
GT199700074A (es) 1998-12-04

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
B11Y Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired