ATE442135T1 - 5ht2c-rezeptor-modulator-zusammensetzungen und anwendungsverfahren - Google Patents

5ht2c-rezeptor-modulator-zusammensetzungen und anwendungsverfahren

Info

Publication number
ATE442135T1
ATE442135T1 AT05855247T AT05855247T ATE442135T1 AT E442135 T1 ATE442135 T1 AT E442135T1 AT 05855247 T AT05855247 T AT 05855247T AT 05855247 T AT05855247 T AT 05855247T AT E442135 T1 ATE442135 T1 AT E442135T1
Authority
AT
Austria
Prior art keywords
methods
receptor modulator
5ht2c receptor
modulator compositions
compositions
Prior art date
Application number
AT05855247T
Other languages
English (en)
Inventor
Dominic P Behan
Brian M Smith
Christina Bjenning
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Application granted granted Critical
Publication of ATE442135T1 publication Critical patent/ATE442135T1/de

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Liquid Crystal Substances (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cosmetics (AREA)
  • Steroid Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
AT05855247T 2004-12-23 2005-12-21 5ht2c-rezeptor-modulator-zusammensetzungen und anwendungsverfahren ATE442135T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US63866704P 2004-12-23 2004-12-23
US68890105P 2005-06-08 2005-06-08
PCT/US2005/046654 WO2006071740A2 (en) 2004-12-23 2005-12-21 5ht2c receptor modulator compositions and methods of use

Publications (1)

Publication Number Publication Date
ATE442135T1 true ATE442135T1 (de) 2009-09-15

Family

ID=36615431

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05855247T ATE442135T1 (de) 2004-12-23 2005-12-21 5ht2c-rezeptor-modulator-zusammensetzungen und anwendungsverfahren

Country Status (25)

Country Link
US (4) US8153621B2 (de)
EP (3) EP2111859A1 (de)
JP (1) JP4886700B2 (de)
KR (3) KR101426850B1 (de)
CN (3) CN102631349A (de)
AT (1) ATE442135T1 (de)
AU (1) AU2005322183B2 (de)
BR (1) BRPI0515862A2 (de)
CA (1) CA2588941A1 (de)
CY (1) CY1109629T1 (de)
DE (1) DE602005016601D1 (de)
DK (1) DK1833473T3 (de)
EA (2) EA201100129A1 (de)
ES (1) ES2331656T3 (de)
HK (1) HK1102766A1 (de)
HR (1) HRP20090641T1 (de)
IL (2) IL183565A0 (de)
NZ (2) NZ589951A (de)
PL (1) PL1833473T3 (de)
PT (1) PT1833473E (de)
RS (1) RS50997B (de)
SG (1) SG158168A1 (de)
SI (1) SI1833473T1 (de)
WO (1) WO2006071740A2 (de)
ZA (1) ZA200705165B (de)

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US7674776B2 (en) 1999-06-14 2010-03-09 Vivus, Inc. Combination therapy for effecting weight loss and treating obesity
US6953787B2 (en) 2002-04-12 2005-10-11 Arena Pharmaceuticals, Inc. 5HT2C receptor modulators
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CN102321023A (zh) 2004-12-21 2012-01-18 艾尼纳制药公司 (r)-8-氯-1-甲基-2,3,4,5-四氢-1h-3-苯并氮杂卓盐酸盐的晶型
ATE442135T1 (de) 2004-12-23 2009-09-15 Arena Pharm Inc 5ht2c-rezeptor-modulator-zusammensetzungen und anwendungsverfahren
JP5249031B2 (ja) 2005-09-01 2013-07-31 イーライ リリー アンド カンパニー ５−ＨＴ２Ｃ受容体アゴニストとしての６−Ｎ結合型へテロ環置換された２，３，４，５−テトラヒドロ−１Ｈ−ベンゾ［ｄ］アゼピン
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AU2010249472B2 (en) * 2009-05-22 2015-09-10 AbbVie Deutschland GmbH & Co. KG Modulators of 5-HT receptors and methods of use thereof
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US9045431B2 (en) 2010-06-02 2015-06-02 Arena Pharmaceuticals, Inc. Processes for the preparation of 5-HT2C receptor agonists
AU2011296033A1 (en) 2010-09-01 2013-04-04 Arena Pharmaceuticals, Inc. Non-hygroscopic salts of 5-HT2C agonists
EP2611781A1 (de) * 2010-09-01 2013-07-10 Arena Pharmaceuticals, Inc. Schnelllösliche darreichungsformen von 5-ht2c-agonisten
EP2611427B1 (de) 2010-09-01 2018-10-17 Arena Pharmaceuticals, Inc. Darreichungsformen von 5-ht2c-agonisten mit modifizierter freisetzung für gewichtskontrolle
CA2808909A1 (en) 2010-09-01 2012-03-08 Arena Pharmaceuticals, Inc. Salts of lorcaserin with optically active acids
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EP2939677A1 (de) * 2010-09-01 2015-11-04 Arena Pharmaceuticals, Inc. Verabreichung von lorcaserin an personen mit nierenerkrankungen
AR088670A1 (es) 2012-10-09 2014-06-25 Arena Pharm Inc Metodo de control del peso
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NZ589951A (en) 2012-11-30
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IL238479A0 (en) 2015-06-30
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US20120252786A1 (en) 2012-10-04
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US20090197868A1 (en) 2009-08-06
EP2322162A1 (de) 2011-05-18
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