AR201730A1 - Procedimiento para la preparacion de nuevos esteres de alfaaminopenicilinas - Google Patents

Procedimiento para la preparacion de nuevos esteres de alfaaminopenicilinas

Info

Publication number: AR201730A1
Authority: AR; Argentina
Prior art keywords: alphaaminopenicillin; esters; procedure; preparation; new
Prior art date: 1970-09-17

Application number

AR241427A

Other languages

English (en)

Spanish (es)

Original Assignee

Astra Laekemedel Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1970-09-17

Filing date

1972-04-12

Publication date

1975-04-15

1970-09-17 Priority claimed from SE7012688A external-priority patent/SE374747B/xx

1970-11-20 Priority claimed from SE7015720A external-priority patent/SE380806B/xx

1972-04-12 Application filed by Astra Laekemedel Ab filed Critical Astra Laekemedel Ab

1975-04-15 Application granted granted Critical

1975-04-15 Publication of AR201730A1 publication Critical patent/AR201730A1/es

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cephalosporin Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

AR241427A 1970-09-17 1972-04-12 Procedimiento para la preparacion de nuevos esteres de alfaaminopenicilinas AR201730A1 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
SE7012688A SE374747B (fi)	1970-09-17	1970-09-17
SE7015720A SE380806B (sv)	1970-11-20	1970-11-20	Forfarande for framstellning av nya estrar av alfa-aminopenicilliner

Publications (1)

Publication Number	Publication Date
AR201730A1 true AR201730A1 (es)	1975-04-15

Family

ID=26655897

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AR241427A AR201730A1 (es)	1970-09-17	1972-04-12	Procedimiento para la preparacion de nuevos esteres de alfaaminopenicilinas
AR258235A AR210991A1 (es)	1970-09-17	1975-04-08	Bencilpenicilanato de 1-etoxicarboniloxietilo para su exclusiva utilizacion como intermediario.

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
AR258235A AR210991A1 (es)	1970-09-17	1975-04-08	Bencilpenicilanato de 1-etoxicarboniloxietilo para su exclusiva utilizacion como intermediario.

Country Status (21)

Country	Link
US (2)	US3873521A (fi)
JP (2)	JPS5317597B1 (fi)
AR (2)	AR201730A1 (fi)
AT (2)	AT309681B (fi)
BE (1)	BE772723A (fi)
BR (1)	BR7106116D0 (fi)
CA (2)	CA960211A (fi)
CH (5)	CH583239A5 (fi)
CS (2)	CS187312B2 (fi)
DD (1)	DD94815A5 (fi)
DK (6)	DK132759C (fi)
ES (3)	ES395145A1 (fi)
FI (4)	FI55203C (fi)
FR (1)	FR2106578B1 (fi)
GB (1)	GB1363506A (fi)
HU (1)	HU165868B (fi)
IE (1)	IE35642B1 (fi)
IT (1)	IT1049876B (fi)
NL (3)	NL164860C (fi)
NO (4)	NO140931C (fi)
SU (2)	SU553936A3 (fi)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1426869A (en) *	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
GB1425933A (en) *	1972-03-13	1976-02-25	Astra Laekemedel Ab	Cephalosporins
US4089963A (en) *	1972-03-13	1978-05-16	Astra Pharmaceutical Products, Inc.	Esters of amidinopenicillanic acids, pharmaceutical preparations and method for treating infectious diseases
GB1437088A (en) *	1972-05-25	1976-05-26	Beecham Group Ltd	Esters of penicillins and cephalosporins
NL7401782A (fi) *	1973-02-14	1974-08-16
GB1550359A (en) *	1975-08-07	1979-08-15	Beecham Group Ltd	Antibiotic compositions for oral administration
US4247461A (en) *	1979-11-16	1981-01-27	Bristol-Myers Company	Esterification process using methoxymethyl-P-toluenesulfonate
US4340539A (en) *	1980-01-21	1982-07-20	Bristol-Myers Company	Derivatives of 6-bromo penicillanic acid
CA1212105A (en)	1980-04-30	1986-09-30	Shoji Ikeda	Ampicillin esters and production thereof
FR2482587A1 (fr) *	1980-05-14	1981-11-20	Poudres & Explosifs Ste Nale	Procede de synthese de chloroformiates a-chlores et nouveaux chloroformiates a-chlores
US4321253A (en) *	1980-08-22	1982-03-23	Beatty Morgan L	Suspension of microencapsulated bacampicillin acid addition salt for oral, especially pediatric, administration
US4479947A (en) *	1981-07-13	1984-10-30	Merck & Co., Inc.	Oral absorption enhancement of carboxylic acid pharmaceuticals using (5-alkyl-2-oxo-1,3-dioxolen-4-yl)methyl ester group
CA1202617A (en) *	1982-03-19	1986-04-01	Norman B. Jones	Bacampicillin napsylate
FR2532933B1 (fr) *	1982-06-29	1987-11-13	Astra Laekemedel Ab	Perfectionnements apportes a la preparation d'antibiotiques
SE454879B (sv) *	1982-06-29	1988-06-06	Astra Laekemedel Ab	Alfa-bromodietylkarbonat samt dess anvendning som mellanprodukt vid framstellning av penicillin g
GB2123821B (en) *	1982-06-29	1987-04-23	Astra Laekemedel Ab	At-halogeno diethyl carbonates and their use in the preparation of antibiotics
IT1190897B (it) *	1982-06-29	1988-02-24	Opos Biochimica Srl	Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
JPS5927900A (ja) *	1982-08-09	1984-02-14	Wakunaga Seiyaku Kk	固定化オリゴヌクレオチド
US4606865A (en) *	1982-09-20	1986-08-19	Astra Lakemedel Aktiebolag	Methods for the preparation of α-bromodiethylcarbonate
DK149079C (da) *	1982-10-06	1986-06-23	Novo Industri As	Fremgangsmaade til fremstilling af et immobiliseret enzympraeparat
IL67637A0 (en) *	1983-01-07	1983-05-15	Orvet Bv	Preparation of 1'-ethoxycarbonyl-oxyethyl esters of penicillins and novel intermediates
IL67177A (en) *	1982-11-04	1985-08-30	Orvet Bv	1-bromoethyl ethyl carbonate,methods for its preparation and 1-bromoethylchloroformate and 1-bromoethylbromoformate obtained as intermediates
IL67445A (en) *	1982-12-09	1985-11-29	Teva Pharma	Ethoxycarbonyloxy ethyl esters of non-steroidal anti-inflammatory carboxylic acids
FR2551058B1 (fr) *	1983-08-26	1986-09-26	Poudres & Explosifs Ste Nale	Procede de preparation de chloroformiates a-chlores
SE8405611D0 (sv) *	1984-11-09	1984-11-09	Astra Laekemedel Ab	Process for stabilization of bacampicillin hydrochloride
US4855455A (en) *	1988-01-22	1989-08-08	W. R. Grace & Co.-Conn.	Preparation of amino acid derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR1021654A (fr) *	1949-07-07	1953-02-23	Lphivens Kemiske Fabrik Ved A	Procédé de production d'éthers-sels aminés de pénicilline et de composés qui s'y rattachent
GB1241844A (en) *	1968-08-23	1971-08-04	Beecham Group Ltd	Penicillins
US3697507A (en) *	1968-09-26	1972-10-10	Leo Pharm Prod Ltd	Esters of {60 -aminobenzylpenicillin
US3660575A (en) *	1968-09-26	1972-05-02	Leo Pharm Prod Ltd	Esters of alpha-aminobenzylpenicillin in dosage unit form

1971
- 1971-09-07 US US178426A patent/US3873521A/en not_active Expired - Lifetime
- 1971-09-14 AT AT795771A patent/AT309681B/de not_active IP Right Cessation
- 1971-09-14 FR FR7133107A patent/FR2106578B1/fr not_active Expired
- 1971-09-14 SU SU1696133A patent/SU553936A3/ru active
- 1971-09-14 AT AT537872A patent/AT311557B/de not_active IP Right Cessation
- 1971-09-15 FI FI2580/71A patent/FI55203C/fi active
- 1971-09-15 GB GB4309071A patent/GB1363506A/en not_active Expired
- 1971-09-15 IE IE1167/71A patent/IE35642B1/xx unknown
- 1971-09-15 CA CA122,881A patent/CA960211A/en not_active Expired
- 1971-09-15 IT IT28678/71A patent/IT1049876B/it active
- 1971-09-16 CH CH1362371A patent/CH583239A5/xx not_active IP Right Cessation
- 1971-09-16 CS CS716617A patent/CS187312B2/cs unknown
- 1971-09-16 DK DK453871A patent/DK132759C/da not_active IP Right Cessation
- 1971-09-16 NO NO3449/71A patent/NO140931C/no unknown
- 1971-09-16 BR BR6116/71A patent/BR7106116D0/pt unknown
- 1971-09-16 HU HUAA684A patent/HU165868B/hu unknown
- 1971-09-16 CH CH859975A patent/CH577513A5/xx not_active IP Right Cessation
- 1971-09-16 CH CH860075A patent/CH589654A5/xx not_active IP Right Cessation
- 1971-09-16 ES ES195145A patent/ES395145A1/es not_active Expired
- 1971-09-16 CS CS71442A patent/CS187316B2/cs unknown
- 1971-09-17 JP JP7184971A patent/JPS5317597B1/ja active Pending
- 1971-09-17 DD DD157795A patent/DD94815A5/xx unknown
- 1971-09-17 BE BE772723A patent/BE772723A/xx not_active IP Right Cessation
- 1971-09-17 NL NL7112789.A patent/NL164860C/xx not_active IP Right Cessation
1972
- 1972-01-31 NO NO236/72A patent/NO140930C/no unknown
- 1972-04-12 AR AR241427A patent/AR201730A1/es active
- 1972-04-14 ES ES401745A patent/ES401745A1/es not_active Expired
1973
- 1973-03-08 US US05/339,364 patent/US3939270A/en not_active Expired - Lifetime
- 1973-03-27 SU SU731899287A patent/SU1153830A3/ru active
- 1973-10-25 CA CA184,183A patent/CA1008447A/en not_active Expired
1974
- 1974-09-27 DK DK509774A patent/DK509774A/da unknown
- 1974-09-27 DK DK509674A patent/DK150200C/da not_active IP Right Cessation
- 1974-12-19 NO NO74744606A patent/NO142670C/no unknown
- 1974-12-31 FI FI3814/74A patent/FI59600C/fi active
1975
- 1975-01-08 ES ES433637A patent/ES433637A1/es not_active Expired
- 1975-04-08 AR AR258235A patent/AR210991A1/es active
- 1975-06-24 JP JP7921675A patent/JPS5537996B2/ja not_active Expired
- 1975-08-20 DK DK375975A patent/DK375975A/da unknown
1976
- 1976-04-20 CH CH493776A patent/CH613207A5/xx not_active IP Right Cessation
1977
- 1977-09-21 CH CH1155377A patent/CH602745A5/xx not_active IP Right Cessation
- 1977-10-13 FI FI773032A patent/FI57951C/fi not_active IP Right Cessation
1978
- 1978-01-31 NL NL7801086A patent/NL7801086A/xx active Search and Examination
- 1978-12-08 NO NO784144A patent/NO142671C/no unknown
1979
- 1979-04-27 FI FI791386A patent/FI59103C/fi not_active IP Right Cessation
1980
- 1980-03-17 NL NLAANVRAGE8001563,A patent/NL171160C/xx not_active IP Right Cessation
- 1980-03-27 DK DK133380A patent/DK150201C/da not_active IP Right Cessation
1982
- 1982-04-07 DK DK163482A patent/DK158519C/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
BE772723A (fr)	1972-03-17
NO142670B (no)	1980-06-16
FI791386A (fi)	1979-04-27
FI55203C (fi)	1979-06-11
CH583239A5 (fi)	1976-12-31
FI55203B (fi)	1979-02-28
FI59103B (fi)	1981-02-27
ES433637A1 (es)	1976-11-16
NO140931C (no)	1979-12-12
AT309681B (de)	1973-08-27
FI773032A (fi)	1977-10-13
GB1363506A (en)	1974-08-14
DK150200C (da)	1987-07-06
FR2106578A1 (fi)	1972-05-05
CH589654A5 (fi)	1977-07-15
IT1049876B (it)	1981-02-10
JPS5317597B1 (fi)	1978-06-09
CH577513A5 (fi)	1976-07-15
CH613207A5 (fi)	1979-09-14
JPS5136491A (fi)	1976-03-27
NL7112789A (fi)	1972-03-21
NO142670C (no)	1980-09-24
FI59600B (fi)	1981-05-29
DK158519B (da)	1990-05-28
US3873521A (en)	1975-03-25
FI381474A (fi)	1974-12-31
FI57951B (fi)	1980-07-31
DD94815A5 (fi)	1973-01-05
NL164860C (nl)	1981-02-16
CS187312B2 (en)	1979-01-31
NO142671B (no)	1980-06-16
CA960211A (en)	1974-12-31
NO142671C (no)	1980-09-24
DK150201C (da)	1987-07-06
DK150201B (da)	1987-01-05
NO140930C (no)	1979-12-12
NL8001563A (nl)	1980-06-30
DK133380A (da)	1980-03-27
DK509674A (fi)	1975-06-02
CH602745A5 (fi)	1978-07-31
HU165868B (fi)	1974-12-28
DE2144457B2 (de)	1977-05-05
DK375975A (fi)	1975-08-20
BR7106116D0 (pt)	1973-03-20
JPS5537996B2 (fi)	1980-10-01
CS187316B2 (fi)	1979-01-31
CA1008447A (en)	1977-04-12
IE35642B1 (en)	1976-04-14
FI57951C (fi)	1980-11-10
DE2144457A1 (fi)	1972-03-30
DK132759C (da)	1976-07-05
DK163482A (da)	1982-04-07
US3939270A (en)	1976-02-17
IE35642L (en)	1972-03-17
NO140931B (no)	1979-09-03
AR210991A1 (es)	1977-10-14
NO784144L (no)	1972-03-20
NO744606L (fi)	1972-03-20
AT311557B (de)	1973-11-26
SU553936A3 (ru)	1977-04-05
NL171160B (nl)	1982-09-16
NL7801086A (nl)	1978-05-31
FR2106578B1 (fi)	1975-06-06
ES401745A1 (es)	1976-05-16
DK132759B (da)	1976-02-02
NO140930B (no)	1979-09-03
SU1153830A3 (ru)	1985-04-30
DK150200B (da)	1987-01-05
FI59103C (fi)	1981-06-10
FI59600C (fi)	1981-09-10
DK158519C (da)	1990-11-05
ES395145A1 (es)	1974-11-16
DK509774A (fi)	1975-05-26
NL171160C (nl)	1983-02-16

Publication	Publication Date	Title
AR201730A1 (es)	1975-04-15	Procedimiento para la preparacion de nuevos esteres de alfaaminopenicilinas
AR193370A1 (es)	1973-04-23	Procedimiento para la preparacion de inhibidores para hidrolasas de glicosidos
AR192303A1 (es)	1973-02-14	Procedimiento para la preparacion de acidos 5-fenil-isoxazol-3-carboxilicos
AR204898A1 (es)	1976-03-19	Procedimiento para la preparacion de nuevos ureidofenoxi-2-hidroxi-3-aminopropanos
AR194205A1 (es)	1973-06-29	Procedimiento para la preparacion de naftilaquilaminas
AR199879A1 (es)	1974-10-08	Procedimiento para la elaboracion de 4-aza-benzimidazoles
AR192582A1 (es)	1973-02-28	Procedimiento para la produccion de acidos 4-oxo-4h-1-benzopiran-2-carboxilicos
AR202376A1 (es)	1975-06-06	Procedimiento para la produccion de nuevas aminofenil-imino-pirrolidinas
AR192765A1 (es)	1973-03-14	Procedimiento para la preparacion de derivados de la fenil-3-tiourea
AR196870A1 (es)	1974-02-28	Procedimiento para la preparacion de 1-oxi- bencimidazoles antihelminticos
AR195786A1 (es)	1973-11-09	Procedimiento para la preparacion de derivados de benzocicloheptaisoquinolina
AR199762A1 (es)	1974-09-30	Procedimiento para la preparacion de 5-fluoro-pirimidinas
AR204899A1 (es)	1976-03-19	Procedimiento para la preparacion de 3-carbamoiloximetilcefalosporinas
AR192783A1 (es)	1973-03-14	Procedimiento para la preparacion de nuevas tioureas
AR199361A1 (es)	1974-08-23	Procedimiento para la preparacion de nuevos esteres basicos
AR200139A1 (es)	1974-10-24	Procedimiento para la preparacion de fenilimidazolidinonas
RO70179A (ro)	1982-10-11	Procedeu pentru prepararea izoprenului
AR194401A1 (es)	1973-07-13	Procedimiento para la preparacion de derivados de kasugamicina
IT1051240B (it)	1981-04-21	Procedimento per la preparazione di zeaxantina
AR202882A1 (es)	1975-07-31	Procedimiento para la fabricacion de derivados de 1-o-carbamoilmetoxifenoxi-3-amino-2-propanol
AR194904A1 (es)	1973-08-24	Procedimiento para la elaboracion de nuevos halogeno-esteroides
AR199892A1 (es)	1974-10-08	Procedimiento para la preparacion de esteres alquilicos de acido-metilquinoseolin-1,4-n-dioxido-2-carboxilico
AR193576A1 (es)	1973-04-30	Procedimiento para la preparacion de pirimidotriacinas
AR199767A1 (es)	1974-09-30	Procedimiento para la preparacion de nuevos 3-guanidino-alquil-tiofenos
AR192565A1 (es)	1973-02-28	Procedimiento para la produccion de oudenona